LT052

Name: LT052
Brand: Adooq Bioscience
SKU: A24429
Rating: 5 (288 reviews)

Catalog No.: A24429

BET BD1 inhibitor

LT052 is a highly selective BET BD1 inhibitor with an IC₅₀ of 87.7 nM. It demonstrates nanomolar potency against BRD4 BD1 and exhibits 138-fold selectivity over BRD4 BD2 (IC₅₀ = 12.130 μM). LT052 possesses anti-inflammatory activity and is applicable in acute gout arthritis research.

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Grouped product items
Size	Price	Stock
5mg	$72.00	In stock
10mg	$124.00	In stock
50mg	$368.00	In stock
100mg	$720.00	In stock
Bulk Size	Bulk Discount

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Biological Activity

Description	LT052 is a highly selective BET BD1 inhibitor with an IC₅₀ of 87.7 nM. It demonstrates nanomolar potency against BRD4 BD1 and exhibits 138-fold selectivity over BRD4 BD2 (IC₅₀ = 12.130 μM). LT052 possesses anti-inflammatory activity and is applicable in acute gout arthritis research.

Product Information

Catalog Num	A24429
Formula	C22H19N5O4S
Molecular Weight	449.48
CAS Number	2543545-44-2
SMILES	O=S(C1=CC=CC=C1OC)(NC2=C3N=C(N4C=C(C)N=C4)C=C5C3=C(N(C)C5=O)C=C2)=O
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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