OARV-771

Name: OARV-771
Brand: Adooq Bioscience
SKU: A24409
Rating: 5 (288 reviews)

Catalog No.: A24409

BET degrader

OARV-771 is a VHL-based BET degrader (PROTAC) with enhanced cell permeability. It exhibits potent degradation activity with DC50 values of 6 nM, 1 nM, and 4 nM for BRD4, BRD2, and BRD3, respectively.

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Grouped product items
Size	Price	Stock
5mg	$585.00	In stock
10mg	$1,008.00	In stock
50mg	$2,990.00	In stock
100mg	$5,850.00	In stock
Bulk Size	Bulk Discount

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Biological Activity

Description	OARV-771 is a VHL-based BET degrader (PROTAC) with enhanced cell permeability. It exhibits potent degradation activity with DC50 values of 6 nM, 1 nM, and 4 nM for BRD4, BRD2, and BRD3, respectively.

Product Information

Catalog Num	A24409
Formula	C49H59ClN8O8S2
Molecular Weight	987.62
CAS Number	2683008-37-7
SMILES	CC1=C(C)SC2=C1C(C3=CC=C(C=C3)Cl)=N[C@@H](CC(OCCOCCCOCC(N[C@@H](C(C)(C)C)C(N4[C@@H](C[C@H](C4)O)C(N[C@H](C5=CC=C(C6=C(C)N=CS6)C=C5)C)=O)=O)=O)=O)C7=NN=C(C)N27
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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