Other Inhibitors

Cat. No.

A13689

CAS No.

229971-81-7

Exherin (ADH-1)

Synonyms: NSC729477; ADH-1

Exherin is a small, cyclic pentapeptide vascular-targeting agent with potential antineoplastic and antiangiogenic activities.

Cat. No.

A11003

CAS No.

65-19-0

Yohimbine hydrochloride

Synonyms: Antagonil; Yohimbe; Aphrodine hydrochloride; Yohimbine monohydrochloride

Yohimbine hydrochloride (Antagonil) is a α2-adrenoceptor antagonist (pKi values are 8.52, 8.00 and 9.17 for human α2A, α2B and α2C receptors respectively)

Cat. No.

A11670

CAS No.

108341-18-0

Noradrenaline bitartrate monohydrate

Synonyms: Levophed

Noradrenaline bitartrate monohydrate (Levophed) is a direct alpha-adrenergic receptors stimulator.

Cat. No.

A12194

CAS No.

256925-03-8

AL082D06

Synonyms: D-06

AL082D06 is a nonsteroidal glucocorticoid receptor antagonist.

Cat. No.

A12355

CAS No.

81486-22-8

Nipradilol

Synonyms: Nipranol; Nipradolol; BRN 3566879

nipradilol is an alpha(1),beta-blocker with a nitric oxide donative action

Cat. No.

A12466

CAS No.

240427-90-1

20-HEDE

Synonyms: WIT 002

20-HEDE (WIT 002) is an antagonist of 20-hydroxyeicosatetraenoic acid (20-HETE).

Cat. No.

A12568

CAS No.

1005491-05-3

Tirasemtiv (CK-2017357)

Synonyms: CK-2017357

Tirasemtiv amplifies skeletal muscle response to nerve activation in humans.

Cat. No.

A12643

CAS No.

125720-84-5

(E)-Alprenoxime

Synonyms: CDDD-1815

(E)-Alprenoxime is the isomer of the Alprenoxime. Alprenoxime is a site-activated ocular β-blocker.

Cat. No.

A12878

CAS No.

1104080-42-3

SNT-207858

SNT207858 is a 22 nM MC4 antagonist with a 170-fold selectivity vs. MC3 and a 40-fold selectivity versus MC5.

Cat. No.

A12908

CAS No.

1420071-30-2

Bioymifi

Bioymifi is a potent and selective small molecule agonist of DR5 that directly targets DR5, specifically binds the ECD of DR5 (Kd ~1.2 μM), and induces the formation of DR5 aggregates and DR5 activation.

Cat. No.

A12913

CAS No.

1370554-01-0

Cilliobrevin D

Ciliobrevin D is the first specific small molecule antagonist of cytoplasmic dynein

Cat. No.

A13124

CAS No.

1064662-40-3

SNT-207707

SNT-207707 is an oral MC4-Receptor Antagonist

Cat. No.

A13178

CAS No.

187269-40-5

Bimosiamose

Synonyms: TBC 1269

Bimosiamose is a pan-selectin antagonist, inhibits E-, P-, and L-selectin with IC50s of 88 μM, 20 μM, and 86 μM, respectively, and can be used in the research of inflammatory disease.

Cat. No.

A13400

CAS No.

14556-46-8

Bupranolol

Synonyms: B 1312; BRN 2272923; Bupranololum; KL 255Ophtorenin

Bupranolol is a non-selective beta blocker without intrinsic sympathomimetic activity (ISA), but with strong membrane stabilizing activity.

Cat. No.

A13919

CAS No.

22273-09-2

Fluorocurarine chloride

Fluorocurarine chloride is a short-acting selective sympathetic ganglioblocker with weak antagonist activity on the nicotinic receptor at the neuromuscular junction.

Cat. No.

A14052

CAS No.

2141977-22-0

YH249

YH249 is the first highly specific, direct p300/β-catenin antagonist.

Cat. No.

A14150

CAS No.

1256037-58-7

TRX 818

TRX-818 is a new, potent and multi-targeted anti-cancer agent in numerous human cancer cell lines.

Cat. No.

A15329

CAS No.

211364-78-2

R18

R18, antagonist of 14.3.3 proteins (KD ??? 80 nM). Competitively inhibits 14.3.3-ligand interactions without requiring phosphorylation.

Cat. No.

A17177

CAS No.

2227996-00-9

EG01377 TFA

Synonyms: EG 01377

EG01377 TFA salt is a selective neuropilin-1 (NRP1) antagonist. CAS: 2227996-00-9 (Free base)

Cat. No.

A17588

CAS No.

1188-38-1

Carglumic Acid

Synonyms: OE312; AJ 266447; AJ-26647; Carglumic Acid.

Carglumic acid (N-Carbamyl-L-glutamic acid), a functional analogue of N-acetylglutamate (NAG) and a carbamoyl phosphate synthetase 1 (CPS1) activator, is used to treat acute and chronic hyperammonemia associated with NAG synthase (NAGS) deficiency.

Cat. No.

A18152

CAS No.

23642-66-2

Benfluorex hydrochloride

Synonyms: Benfluorex HCl; Lipophoral; Mediator; JP 992; EINECS 245-801-8; Mediaxal; Balans

Benfluorex hydrochloride (JP-992 hydrochloride) is a hepatic nuclear factor 4 alpha (HNF4α) activator.

Cat. No.

A19055

CAS No.

421581-52-4

G6PD activator AG1

G6PD activator AG1 is a glucose-6-phosphate dehydrogenase (G6PD) activator with an EC50 of 3 μ, extracted from patent WO2019023264A1, compound AG1.

Cat. No.

A19359

CAS No.

439685-79-7

Pro-xylane

Synonyms: Hydroxypropyl tetrahydropyrantriol

Pro-xylane (Hydroxypropyl tetrahydropyrantriol) is a biologically active C-glycoside in aqueous media, acts as an activator of glycosaminoglycans (GAGs) biosynthesis.

Cat. No.

A19478

CAS No.

6266-66-6

PEO-IAA

Synonyms: 2-(1H-Indol-3-yl)-4-oxo-4-phenyl-butyric acid

PEO-IAA is an indole-3-acetic acid (IAA) antagonist. PEO-IAA is an auxin antagonist that binds to transport inhibitor response 1/auxin signaling F-box proteins (TIR1/AFBs).

Cat. No.

A19489

CAS No.

81921-35-9

N6-Methyladenosine 5'-monophosphate disodium salt

N6-Methyladenosine 5'-monophosphate disodium salt is an activator of glycogen phosphorylase b, with a Ka value of 22 µM. N6-Methyladenosine 5'-monophosphate disodium salt is a non-competitive rat adenylate kinase II inhibitor.