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Zavabresib

Catalog No.: A40314
BET Inhibitor
Zavabresib is a potent inhibitor of bromodomain and extraterminal domain (BET) proteins. It exhibits significant anticancer activity, particularly in prostate cancer, demonstrated by IC50 values of 0.043 and 0.034 μM against LNCaP and 22Rv1 cell lines, respectively. This compound is a valuable tool for investigating the role of BET inhibition in cancer biology and therapeutic development.
Zavabresib 2089390-09-8 BET Inhibitor
Grouped product items
Size Price Stock Qty
5mg
$655.00
In stock
10mg
$1,090.00
In stock
25mg
$2,015.00
In stock
50mg
$2,280.00
In stock
100mg
$2,960.00
In stock
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Free Delivery on orders over $500
Research use only. We do not sell to patients.
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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionZavabresib is a potent inhibitor of bromodomain and extraterminal domain (BET) proteins. It exhibits significant anticancer activity, particularly in prostate cancer, demonstrated by IC50 values of 0.043 and 0.034 μM against LNCaP and 22Rv1 cell lines, respectively. This compound is a valuable tool for investigating the role of BET inhibition in cancer biology and therapeutic development.
Product Information
Catalog NumA40314
FormulaC31H25N5O3
Molecular Weight515.56
CAS Number2089390-09-8
SMILESO=C(C1=CC=C(C2=CN(C(C3=NC=CC=C3)(C)C4=NC=CC=C4)C5=C2N=CC(C6=C(C)ON=C6C)=C5)C=C1)O
SynonymsBET-IN-16
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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