AS703026 (Pimasertib)

Catalog No.: A10089

MEK1/2 inhibitor

AS703026 (Pimasertib) Chemical Structure

CAS NO. 1236699-92-5

AS703026 is a novel, selective, orally bioavailable MEK1/2 inhibitor that inhibits growth and survival of MM cells and cytokine-induced osteoclast differentiation.

Availability: In stock

Package Price Qty
5 mg
$40.00
10 mg
$70.00
50 mg
$180.00
100 mg
$300.00
10mM * 1mL in DMSO
$93.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

AS703026 is a novel, selective, orally bioavailable MEK1/2 inhibitor that inhibits growth and survival of MM cells and cytokine-induced osteoclast differentiation.
In vitro (25°C) DMSO 86 mg/mL (199.44 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 0.5% CMC/0.25% Tween 80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.19 mL 115.96 mL 231.91 mL
0.5 mM 4.64 mL 23.19 mL 46.38 mL
1 mM 2.32 mL 11.6 mL 23.19 mL
5 mM 0.46 mL 2.32 mL 4.64 mL

*The above data is based on the productmolecular weight 431.2 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10089
Actions Inhibitor
M. Wt 431.2
Formula C15H15FIN3O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1236699-92-5
Synonyms AS-703026, MSC1936369B
SMILES C1=CC(=C(C=C1I)F)NC2=C(C=CN=C2)C(=O)NC[[email protected]@H](CO)O

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