EPZ005687

Catalog No.: A12439

EZH2 inhibitor

EPZ005687

EPZ005687 Chemical Structure

CAS NO. 1396772-26-1

EPZ005687 is a potent inhibitor of EZH2 (K(i) of 24 nM)

Availability: In stock

Package Price Qty
5 mg
$60.00
10 mg
$100.00
25 mg
$200.00
50 mg
$350.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

EPZ005687 is a potent inhibitor of EZH2 (K(i) of 24 nM)
Targets
EZH2 (Cell-free assay)
24 nM(Ki)
In vitro DMSO 2 mg/mL (3.7 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.53 mL 92.65 mL 185.3 mL
0.5 mM 3.71 mL 18.53 mL 37.06 mL
1 mM 1.85 mL 9.26 mL 18.53 mL
5 mM 0.37 mL 1.85 mL 3.71 mL

*The above data is based on the productmolecular weight 539.67. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12439
Actions Inhibitor
M. Wt 539.67
Formula C32H37N5O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1396772-26-1
Synonyms EPZ-005687
SMILES CC1=CC(=C(C(=O)N1)CNC(=O)C2=C3C=NN(C3=CC(=C2)C4=CC=C(C=C4)CN5CCOCC5)C6CCCC6)C

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