EZH2-IN-17 is a potent EZH2 inhibitor with an IC50 value of 0.95 nM, demonstrating significant selectivity and oral bioavailability. This compound exhibits robust anti-proliferative activity against various lymphoma cell lines, including WSU-DLCL2, Pfeiffer, and Karpas-422, with IC50 values of 2.36 nM, 1.73 nM, and 1.82 nM, respectively. EZH2-IN-17 is useful for research focused on epigenetic modulation and the investigation of EZH2's role in cancer progression.
EZH2-IN-17 is a potent EZH2 inhibitor with an IC50 value of 0.95 nM, demonstrating significant selectivity and oral bioavailability. This compound exhibits robust anti-proliferative activity against various lymphoma cell lines, including WSU-DLCL2, Pfeiffer, and Karpas-422, with IC50 values of 2.36 nM, 1.73 nM, and 1.82 nM, respectively. EZH2-IN-17 is useful for research focused on epigenetic modulation and the investigation of EZH2's role in cancer progression.
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