HIV Protease

Cat. No.

A11504

CAS No.

159989-64-7

Nelfinavir

Synonyms: Viracept; AG 1341

Nelfinavir is a potent and orally bioavailable human immunodeficiency virus HIV-1 protease inhibitor (Ki=2 nM) and is widely prescribed in combination with HIV reverse transcriptase inhibitors for the treatment of HIV infection.

Cat. No.

A11378

CAS No.

127779-20-8

Saquinavir

Saquinavir is a protease inhibitor. Proteases are enzymes that cleave protein molecules into smaller fragments. Saquinavir inhibits both HIV-1 and HIV-2 proteases.

Cat. No.

A11985

CAS No.

161814-49-9

Amprenavir

Amprenavir is an human immunodeficiency virus (HIV) protease inhibitor with IC50 of 14.6 ± 12.5 ng/ml for wild-type HIV isolates

Cat. No.

A10096

CAS No.

229975-97-7

Atazanavir sulfate (BMS-232632-05)

Synonyms: CGP-73547; Reyataz; Zrivada; BMS-232632-05

Atazanavir is an antiretroviral drug of the protease inhibitor (PI) class. Like other antiretrovirals, it is used to treat infection of human immunodeficiency virus (HIV).

Cat. No.

A10097

CAS No.

198904-31-3

Atazanavir

Synonyms: Reyataz; BMS232632

Atazanavir is an antiretroviral drug of the protease inhibitor (PI) class. Like other antiretrovirals, it is used to treat infection of human immunodeficiency virus (HIV).

Cat. No.

A10537

CAS No.

192725-17-0

Lopinavir (ABT-378)

Synonyms: ABT-378

Lopinavir is an inhibitor of the HIV protease.

Cat. No.

A10799

CAS No.

155213-67-5

Ritonavir

Synonyms: Norvir; Norvir Softgel

Ritonavir is a protease inhibitor with activity against Human Immunodeficiency Virus Type 1 (HIV-1). Protease inhibitors block the part of HIV called protease.Ritonavir inhibits the HIV viral proteinase enzyme which prevents cleavage of the gag-pol polyprotein, resulting in noninfectious, immature viral particles.

Cat. No.

A11201

CAS No.

357263-13-9

BMS-806 (BMS 378806)

Synonyms: BMS378806

BMS-806, also known as BMS-378806 , is a type of medicine called an entry inhibitor. Entry inhibitors work by blocking HIV from entering human cells. BMS-378806 (BMS-806) is a small molecule that blocks the binding of host-cell CD4 with viral gp120 protein and therefore inhibits the first steps of HIV-1 infection.

Cat. No.

A11509

CAS No.

333352-59-3

NBD-557

NBD-557 is a potentially HIV-1 inhibitor.

Cat. No.

A11570

CAS No.

149845-06-7

Saquinavir Mesylate

Synonyms: Ro 31-8959/003

Saquinavir mesylate is an HIV Protease Inhibitor used in antiretroviral therapy.

Cat. No.

A11853

CAS No.

635728-49-3

Darunavir Ethanolate

Synonyms: Prezista; TMC114

Darunavir Ethanolate (Prezista) is an HIV protease inhibitor.

Cat. No.

A11871

CAS No.

157810-81-6

Indinavir sulfate

Synonyms: Crixivan

Indinavir sulfate is a novel hydroxyaminopentane amide class of HIV-1 protease inhibitors.

Cat. No.

A12583

CAS No.

226700-79-4

Fosamprenavir

Synonyms: Gw433908; Aids082186; Amprenavir phosphate

Fosamprenavir is a prodrug of amprenavir, an inhibitor of human immunodeficiency virus (HIV) protease.

Cat. No.

A12980

CAS No.

431980-38-0

RN-18

RN-18 is a HIV-1 viral infectivity factor (HIV-1 Vif) inhibitor with an IC50 of 6 μM in nonpermissive H9 cells.

Cat. No.

A13199

CAS No.

149488-17-5

Trovirdine

Synonyms: LY300046

Trovirdine inhibits HIV-1 RT with an IC50 of 7 nM when employing heteropolymeric primer/template (oligo-DNA/ribosomal RNA)and dGTP as substrate.

Cat. No.

A13598

CAS No.

166335-18-8

PNU-103017

PNU-103017 is an HIV protease inhibitor.

Cat. No.

A14259

CAS No.

159989-65-8

Nelfinavir Mesylate

Nelfinavir Mesylate is a potent HIV protease inhibitor with Ki of 2 nM.

Cat. No.

A15026

CAS No.

864953-39-9

BMS-663068 Tris

Synonyms: BMS663068 (Tris)

BMS-663068 tris is an HIV-1 attachment inhibitor in development for the treatment of HIV-1 infection.

Cat. No.

A15089

CAS No.

226700-81-8

Fosamprenavir Calcium Salt

Synonyms: GW 433908G; Lexiva

Fosamprenavir Calcium Salt is a phosphate ester prodrug of the antiretroviral protease inhibitor amprenavir, with improved solubility over the parent molecule and a potential for reduced pill burden on current dosing regimens; GW433908G is the calcium salt of the prodrug.

Cat. No.

A15262

CAS No.

174484-41-4

Tipranavir

Tipranavir, a nonpeptidic HIV protease inhibitor (NPPI), inhibits the enzymatic activity and dimerization of HIV-1 protease, exerts potent activity against multi-PI-resistant HIV-1 isolates.

Cat. No.

A15825

CAS No.

159519-65-0

Enfuvirtide Acetate(T-20)

Synonyms: Fuzeon; DP178

Enfuvirtide Acetate (T-20) is a 36 amino acid peptide corresponding to a region of gp41, the transmembrane subunit of HIV-1 envelope protein.

Cat. No.

A15965

CAS No.

1443461-21-9

GSK2838232-isomer

Synonyms: GSK-2838232

GSK2838232-isomer is a novel human immune virus (HIV) maturation inhibitor being developed for the treatment of chronic HIV infection.

Cat. No.

A16024

CAS No.

1416258-16-6

(±)-BI-D

(±)-BI-D is a potent ALLINI(An allosteric IN inhibitor) that binds integrase at the LEDGF/p75 binding site.

Cat. No.

A16912

CAS No.

1258453-75-6

ABX-464

Synonyms: SPL-464

ABX-464, also known as SPL-464, is an inhibitor of the HIV replication potentially for the treatment of HIV infection.

Cat. No.

A17178

CAS No.

1392312-45-6

GSK3532795

Synonyms: BMS955176

GSK3532795, also known as BMS-955176, is a potent, orally active, second-generation HIV-1 maturation inhibitor. CAS: 1392312-45-6 (free base) 2023808-13-9 (HCl) 2023798-97-0 (HCl hydrate) 2097784-79-5 (oxalate)