P005091

Catalog No.: A13277

DUB/USP7 Inhibitor

P005091

P005091 Chemical Structure

CAS NO. 882257-11-6

P005091 is a selective inhibitor of ubiquitin-specific protease (USP) 7 (IC50 = 4.2 uM).

Availability: In stock

Package Price Qty
10 mg
$80.00
25 mg
$170.00
50 mg
$250.00
10mM * 1mL in DMSO
$89.00
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Biological Activity

P005091 is a selective inhibitor of ubiquitin-specific protease (USP) 7 (IC50 = 4.2 uM).
Targets
Target Value
USP7EC504.2μM
Calpain1EC50>100μM
MMP13EC50>100μM
CathepsinDEC50>100μM
EKLEC50>100μM
PLA2EC50>100μM
USP2cEC50>100μM
USP5EC50>100μM
USP8cEC50>100μM
USP15EC50>100μM
USP20EC50>100μM
USP21EC50>100μM
USP28EC50>100μM
UCH-L1EC50>100μM
Caspase-3EC50>100μM
CathepsinKEC50>100μM
In vitro (25°C) DMSO 28 mg/mL (80.4 mM)
Water Insoluble
Ethanol Insoluble
In vivo 4% DMSO+30% PEG 400+ddH2O 4 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 28.72 mL 143.59 mL 287.17 mL
0.5 mM 5.74 mL 28.72 mL 57.43 mL
1 mM 2.87 mL 14.36 mL 28.72 mL
5 mM 0.57 mL 2.87 mL 5.74 mL

*The above data is based on the productmolecular weight 348.22. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13277
Actions Inhibitor
CAS No. 882257-11-6
Formula C12H7Cl2NO3S2
M. Wt 348.22
Purity >98%
Synonyms P5091
SMILES CC(=O)C1=CC(=C(S1)SC2=C(C(=CC=C2)Cl)Cl)[N+](=O)[O-]
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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