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TAK-981
Catalog No. A20002 SUMO inhibitorTAK-981 is a first in class and selective inhibitor of the SUMOylation enzymatic cascade, with potential immune-activating and antineoplastic activities. Learn More -
PYR-41
Catalog No. A13254 Ubiquitin E1 InhibitorPYR-41 is a cell-permeable, irreversible ubiquitin-activating enzyme (E1) inhibitor (IC50 < 10 μM). Learn More -
N106
Catalog No. A16183 SUMO-activating enzyme activatorN106, activator of SUMO-activating enzyme, E1 ligase. Increases SERCA2a SUMOylation and activity, and enhances contractility in rat cardiomyocytes in vitro. Learn More -
2-D08
Catalog No. A16852 SUMO inhibitor2-D08 is a cell permeable, mechanistically unique inhibitor of protein sumoylation. It is also inhibits Axl, IRAK4, ROS1, MLK4, GSK3β, RET, KDR and PI3Kα with IC50 values of 0.49, 3.9, 5.3, 9.8, 11, 11, 17 and 35 nM respectively in biochemical assays. Learn More -
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COH000
Catalog No. A17122 SUMO E1 InhibitorCOH000 is a highly specific covalent allosteric SUMO E1 inhibitor with an IC50 of 0.2 μM for SUMOylation in vitro. Learn More -
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