DYRK

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  1. LDN-192960 hydrochloride

    Catalog No. A21390
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    DYRK2 inhibitor
    LDN-192960 hydrochloride is an inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) with IC50s of 10 nM and 48 nM, respectively. Learn More
  2. EHT 5372

    Catalog No. A12586
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    DYRK inhibitor
    EHT 5372 is a strong inhibitor of DYRK??s family kinases, with IC50s of 0.22, 0.28 nM for DYRK1A and DYRK1B, respectively. Learn More
  3. sAJM589

    Catalog No. A18429
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    Myc inhibitor
    sAJM589 is a Myc inhibitor which potently disrupts the Myc-Max heterodimer with an IC50 of 1.8 μM. Learn More
  4. 10074-G5

    Catalog No. A17169
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    c-Myc Inhibitor
    10074-G5 is a c-Myc inhibitor by inhibiting c-Myc/Max heterodimer formation and inhibiting its transcriptional activity with IC50 value of 146 μM. Learn More
  5. ML327

    Catalog No. A17009
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    MYC inhibitor
    ML327 is a blocker of MYC. ML327 mediated transcriptional de-repression of E-cadherin and inhibition of epithelial-to-mesenchymal transition. Learn More
  6. KJ Pyr 9

    Catalog No. A16324
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    MYC inhibitor
    KJ Pyr 9 is a novel small-molecule inhibitor of MYC, KJ-Pyr-9, from a Krhnke pyridine library. Learn More
  7. 10058-F4

    Catalog No. A13725
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    c-Myc-Max inhibitor
    10058-F4 is a c-Myc inhibitor that prevents c-Myc/Max dimerization. Learn More
  8. Mirk-IN-1

    Catalog No. A16255
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    Dyrk1B inhibitor
    Mirk-IN-1 is a potent inhibitor of Dyrk1B(Mirk kianse) and Dyrk1A with IC50 of 68±48 nM and 22±8 nM respectively. Learn More
  9. AZ191

    Catalog No. A14314
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    DYRK inhibitor
    AZ191 is a potent and selective DYRK1B inhibitor with IC50 of 17 nM, about 5- and 110-fold selectivity over DYRK1A and DYRK2. Learn More
  10. ID 8

    Catalog No. A12922
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    DYRK inhibitor
    ID-8 is a DYRK inhibitor. ID 8 also stimulates proliferation at a steady rate (observed in serum-free media supplemented with 10 μM over a 30 day period). Learn More
  11. NU 6102

    Catalog No. A12438
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    CDK inhibitor
    NU6102 is selective for CDK1 and CDK2 compared to CDK4/D1 (IC50=1.6 μM), DYRK1A (IC50=0.9 μM), PDK1 (IC50=0.8 μM) and ROCKII (IC50=0.6 μM). Learn More

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