DYRK

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  1. EHT 5372

    Catalog No. A12586
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    DYRK inhibitor
    EHT 5372 is a strong inhibitor of DYRK??s family kinases, with IC50s of 0.22, 0.28 nM for DYRK1A and DYRK1B, respectively. Learn More
  2. LDN-192960 hydrochloride

    Catalog No. A21390
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    DYRK2 inhibitor
    LDN-192960 hydrochloride is an inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) with IC50s of 10 nM and 48 nM, respectively. Learn More
  3. GSK-626616

    Catalog No. A19273
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    DYRK3 inhibitor
    GSK-626616 is a potent, orally bioavailable inhibitor of DYRK3 (IC50=0.7 nM). Learn More
  4. Paprotrain

    Catalog No. A20346
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    MKLP-2 inhibitor
    Paprotrain is a cell-permeable inhibitor of the kinesin MKLP-2, inhibits the ATPase activity of MKLP-2 with an IC50 of 1.35 μM and a Ki of 3.36 μM and shows a moderate inhibition activity on DYRK1A with an IC50 of 5.5 μM. Learn More
  5. ID 8

    Catalog No. A12922
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    DYRK inhibitor
    ID-8 is a DYRK inhibitor. ID 8 also stimulates proliferation at a steady rate (observed in serum-free media supplemented with 10 μM over a 30 day period). Learn More
  6. AZ191

    Catalog No. A14314
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    DYRK inhibitor
    AZ191 is a potent and selective DYRK1B inhibitor with IC50 of 17 nM, about 5- and 110-fold selectivity over DYRK1A and DYRK2. Learn More
  7. Mirk-IN-1

    Catalog No. A16255
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    Dyrk1B inhibitor
    Mirk-IN-1 is a potent inhibitor of Dyrk1B(Mirk kianse) and Dyrk1A with IC50 of 68±48 nM and 22±8 nM respectively. Learn More
  8. LDN-192960

    Catalog No. A21546
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    DYRK2 inhibitor
    LDN-192960 is an inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) with IC50s of 10 nM and 48 nM, respectively. Learn More

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