CGRP Receptor
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CGRP 8-37 (human)
Catalog No. A16949 CGRP receptor antagonistHCGRP-(8-37) is a human calcitonin gene-related peptide (hCGRP) fragment and also an antagonist of CGRP receptor. Sequence: Val-Thr-His-Arg-Leu-Ala-Gly-Leu-Leu-Ser-Arg-Ser-Gly-Gly-Val-Val-Lys-Asn-Asn-Phe-Val-Pro-Thr-Asn-Val-Gly-Ser-Lys-Ala-Phe ;VTHRLAGLLSRSGGVVKNNFVPTNVGSKAF . Learn More -
Olcegepant
Catalog No. A11512 CGRP1 receptorOlcegepant is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP. Learn More -
Ubrogepant
Catalog No. A21670 CGRP antagonistUbrogepant (MK-1602) is a novel oral calcitonin gene-related peptide receptor (CGRP) antagonist in development for acute treatment of migraine. Learn More -
Olcegepant hydrochloride
Catalog No. A21900 CGRP1 receptor antagonistOlcegepant hydrochloride is the first potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP. Learn More -
MK 3207 HCl
Catalog No. A10598 CGRP Receptor antagonistMK 3207 hydrochloride is a potent CGRP receptor antagonist with IC50 of 0.12 nM. Learn More -
MK-0974 (Telcagepant)
Catalog No. A11255 CGRP receptor antagonistMK-0974 (Telcagepant) is a potent and selective antagonist of the human and rhesus CGRP receptors. Learn More -
BMS-927711
Catalog No. A13102 CGRP receptor antagonistBMS-927711 is a potent, selective, competitive human calcitonin gene-related peptide (CGRP) receptor antagonist that has shown in vivo efficacy without vasoconstrictor effect. Learn More -
MK-3207
Catalog No. A15165 CGRP Receptor antagonistMK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC50= 0.12 nM; Ki value= 0.024 nM); highly selective versus human AM1, AM2, CTR, and AMY3. Learn More