MK 3207 HCl

Catalog No.: A10598

CGRP Receptor antagonist

MK 3207 HCl

MK 3207 HCl Chemical Structure

CAS NO. 957116-20-0

MK 3207 hydrochloride is a potent CGRP receptor antagonist with IC50 of 0.12 nM.

Availability: In stock

Package Price Qty
5 mg
$120.00
10 mg
$230.00
50 mg
$680.00
100 mg
$1,200.00
10mM * 1mL in DMSO
$183.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Marlene Dallmayer, .et al. Targeting the CALCB/RAMP1-axis inhibits growth of Ewing sarcoma, bioRxiv, 2018, 2018

Biological Activity

MK 3207 hydrochloride is a potent CGRP receptor antagonist with IC50 of 0.12 nM.
Targets
CGRP
0.12 nM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.83 mL 84.16 mL 168.32 mL
0.5 mM 3.37 mL 16.83 mL 33.66 mL
1 mM 1.68 mL 8.42 mL 16.83 mL
5 mM 0.34 mL 1.68 mL 3.37 mL

*The above data is based on the productmolecular weight 594.1. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10598
Actions Antagonist
CAS No. 957116-20-0
Formula C31H30ClF2N5O3
M. Wt 594.1
Purity >98%
Synonyms MK3207, MK-3207
SMILES C1CCC2(C1)C(=O)N([[email protected]@H](CN2)C3=CC(=CC(=C3)F)F)CC(=O)NC4=CC5=C(C[[email protected]@]6(C5)C7=C(NC6=O)N=CC=C7)C=C4.Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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