Black Friday & Year End Sale starting Nov 21st 2022 through Jan 2nd 2023, enjoy 20% off sitewide

MK-0974 (Telcagepant)

Catalog No.: A11255

CGRP receptor antagonist

MK-0974 (Telcagepant)

MK-0974 (Telcagepant) Chemical Structure

CAS NO. 781649-09-0

MK-0974 (Telcagepant) is a potent and selective antagonist of the human and rhesus CGRP receptors.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $175.00

Special Price $140.00

10 mg

Regular Price: $300.00

Special Price $240.00

25 mg

Regular Price: $550.00

Special Price $440.00

50 mg

Regular Price: $900.00

Special Price $720.00

Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

MK-0974 (Telcagepant) is a potent and selective antagonist of the human and rhesus CGRP receptors.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.65 mL 88.26 mL 176.52 mL
0.5 mM 3.53 mL 17.65 mL 35.3 mL
1 mM 1.77 mL 8.83 mL 17.65 mL
5 mM 0.35 mL 1.77 mL 3.53 mL

*The above data is based on the productmolecular weight 566.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11255
Actions Antagonist
CAS No. 781649-09-0
Formula C26H27F5N6O3
M. Wt 566.5
Purity >98%
Synonyms Telcagepant
SMILES C1C[[email protected]](C(=O)N(C[[email protected]@H]1C2=C(C(=CC=C2)F)F)CC(F)(F)F)NC(=O)N3CCC(CC3)N4C5=C(NC4=O)N=CC=C5

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy MK-0974 (Telcagepant) | MK-0974 (Telcagepant) Supplier | purchase | cost | manufacturer | order | distributor | buy 781649-09-0| 781649-09-0 Supplier | purchase 781649-09-0 | 781649-09-0 cost | 781649-09-0 manufacturer | order 781649-09-0 | 781649-09-0 distributor