Name: BioE-1115
SKU: A22301
Price: 162 USD
Rating: 5 (288 reviews)

Catalog No.

Product Name

Application

Product Information

Product Citation

A13153

WNK-IN-11

WNK inhibitor

WNK-IN-11 is an allosteric With-No-Lysine (WNK) kinase inhibitor, with an IC50 of 4 nM for WNK1.

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A13188

SRPIN340

SRPK inhibitor

SRPIN340 is a cell-permeable isonicotinamide that acts as an ATP-competitive SRPK1-selective inhibitor (IC50 = 0.14 and 1.8 μM, respectively, against mSRPK1 and mSRPK2) with much reduced activity against 143 other kinases.

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A15922

ML-281

STK33 inhibitor

ML-281 is a potent ans selective STK33 inhibitor with IC50 value of 14 nM.

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A16205

WNK463

pan-WNK-kinase inhibitor

WNK463 is an orally bioavailable pan-WNK-kinase inhibitor.

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- Lu DC, .et al. , Pflugers Arch, 2019, Dec;471(11-12):1539-1549 PMID: 31729557
A17120

SGC GAK 1

GAK inhibitor

SGC GAK 1 is a high affinity cyclin G associated kinase (GAK) inhibitor.

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A18395

ZT-12-037-01

ATP-competitive STK19 inhibitor

ZT-12-037-01 is a potent, selective, ATP-competitive STK19 inhibitor. ZT-12-037-01 effectively blocks oncogenic NRAS-driven melanocyte malignant transformation and melanoma growth in vitro and in vivo.

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A18640

SPHINX31

Serine/arginin kinase 1 inhibitor

SPHINX31 is a potent inhibitor of serine/arginine-rich protein kinase 1 (SRPK1; IC50 = 5.9 nM).

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A18656

LP-935509

AAK1 inhibitor

LP-935509 is a potent inhibitor of the Adapter protein-2 Associated Kinase 1 (AAK1).

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A18792

SRPKIN-1

SRPK1/2 inhibitor

SRPKIN-1 is a covalent and irreversible SRPK1/2 inhibitor with IC50s of 35.6 and 98 nM, respectively. Anti-angiogenesis effect.

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A19702

BAY-524

Bub1 inhibitor

BAY-524 is a Bub1 inhibitor, with an IC50 of 450 nM for human Bub1 in the presence of 2 mM ATP.

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A19710

BAY-320

Bub1 inhibitor

BAY-320 is a Bub1 inhibitor, with an IC50 of 680 nM for human Bub1 in the presence of 2 mM ATP.

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A19806

GCN2iB

GCN2 inhibitor

GCN2iB is an ATP-competitive inhibitor of a serine/threonine-protein kinase general control nonderepressible 2 (GCN2), with an IC50 of 2.4 nM.

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A19868

BAY-1816032

BUB1 kinase inhibitor

BAY-1816032 is a potent and oral available BUB1 (budding uninhibited by benzimidazoles 1) kinase inhibitor with an IC50 of 7 nM.

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A19970

2OH-BNPP1

BUB1 kinase inhibitor

2OH-BNPP1 is an inhibitor of BUB1 kinase, a Ser/Thr kinase, used for the treatment of cancer.

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A20412

GCN2-IN-1

GCN2 inhibitor

GCN2-IN-1 (A-92) is a potent general control nonderepressible 2 kinase (GCN2) inhibitor with an IC50 of <0.3 μM in the enzyme assay and an IC50 of 0.3-3 μM in the cell assay.

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A20447

STK16-IN-1

STK16 kinase inhibitor

STK16-IN-1 is a STK16 kinase inhibitor with an IC50 of 295 nM.

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A22301

BioE-1115

PASK inhibitor

BioE-1115 is a highly selective and potent PAS kinase (PASK) inhibitor with an IC50 of ~4 nM. BioE-1115 is also a potent casein kinase 2α inhibitor with an IC50 of ~10 μM.

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Serine/threonine kinase