TRPV

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  1. SB-705498

    Catalog No. A11143
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    TRPV1 antagonist
    SB-705498 is a potent, selective and orally bioavailable TRPV1 antagonist. Learn More
  2. Capsazepine

    Catalog No. A21208
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    TRPV1 receptor
    Capsazepine is a synthetic analogue of the sensory neurone excitotoxin, and an antagonist of TRPV1 receptor with an IC50 of 562 nM. Learn More
  3. SB366791

    Catalog No. A15857
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    TRPV1 receptor antagonist
    SB-366791 is a novel, potent, and selective, cinnamide TRPV1 antagonist. Learn More
  4. Mavatrep

    Catalog No. A15778
    TRPV1 antagonist
    Mavatrep is an orally bioavailable TRPV1 antagonist (Ki=6.5 nM), exhibits minimal effect on the enzymatic activity (IC50 > 25 μM) of CYP isoforms 3A4, 1A2, and 2D6. Learn More
  5. MRS1477

    Catalog No. A15498
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    TRPV1 modulator
    MRS1477 is a TRPV1 positive allosteric modulator. Learn More
  6. Linoleyl ethanolamide

    Catalog No. A15496
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    Linoleylethanolamide is an endocannabinoid that also binds to TRPV1 (Ki = 5.60 uM). Learn More
  7. A-889425

    Catalog No. A13497
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    TRPV1 receptor antagonist
    A-889425 is a selective TRPV1 receptor antagonist. A-889425 blocks TRPV1 channels with an IC50 of 335 nM (rat) and 34 nM (human). Learn More
  8. AMG517

    Catalog No. A12727
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    TRPV1 antagonist
    AMG 517 is a potent and selective TRPV1 antagonist. Learn More
  9. A-1165442

    Catalog No. A21516
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    TRPV1 antagonist
    A-1165442 is a potent, competitive and orally available TRPV1 antagonist with an IC50 of 9 nM for human TRPV1. Learn More
  10. Resiniferatoxin

    Catalog No. A14003
    vanilloid receptor agonist
    Resiniferatoxin is a natural analog of capsaicin (Item No. 92350) isolated from some plants of the genus Euphorbia, including E. resinifera. Learn More
  11. GSK1016790A

    Catalog No. A15854
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    TRPV4 Activator
    GSK1016790A is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34nM in choroid plexus epithelial cells. Learn More
  12. GSK-2193874

    Catalog No. A14201
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    TRPV4 blocker
    GSK2193874 was identified as a selective, orally active TRPV4 blocker that inhibits Ca(2+) influx through recombinant TRPV4 channels and native endothelial TRPV4 currents. Learn More
  13. (+)-Camphor

    Catalog No. A16423
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    Camphor is a waxy, flammable, white or transparent solid with a strong aroma, often used to relieve pain, reduce itching and treat fungal infections. It can activate TRPV1 and TRPV3 Learn More
  14. (Z)-Capsaicin

    Catalog No. A18179
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    TRPV1 agonist
    Zucapsaicin, also known as cis-Capsaicin, is a medication used to treat osteoarthritis of the knee and other neuropathic pain. It is applied three times daily for a maximum of three months. It reduces pain, and improves articular functions. Learn More
  15. JNJ-17203212

    Catalog No. A12766
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    TRPV1 antagonist
    NJ-17203212 is a novel and selective TRPV1 antagonist, with IC50 of 65 nM and 102 nM for human TRPV1 and rat TRPV1. Learn More

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