TRPV

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  1. SB-705498

    Catalog No. A11143
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    TRPV1 antagonist
    SB-705498 is a potent, selective and orally bioavailable TRPV1 antagonist. Learn More
  2. SB366791

    Catalog No. A15857
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    TRPV1 receptor antagonist
    SB-366791 is a novel, potent, and selective, cinnamide TRPV1 antagonist. Learn More
  3. Mavatrep

    Catalog No. A15778
    TRPV1 antagonist
    Mavatrep is an orally bioavailable TRPV1 antagonist (Ki=6.5 nM), exhibits minimal effect on the enzymatic activity (IC50 > 25 μM) of CYP isoforms 3A4, 1A2, and 2D6. Learn More
  4. MRS1477

    Catalog No. A15498
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    TRPV1 modulator
    MRS1477 is a TRPV1 positive allosteric modulator. Learn More
  5. Linoleyl ethanolamide

    Catalog No. A15496
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    Linoleylethanolamide is an endocannabinoid that also binds to TRPV1 (Ki = 5.60 uM). Learn More
  6. A-889425

    Catalog No. A13497
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    TRPV1 receptor antagonist
    A-889425 is a selective TRPV1 receptor antagonist. A-889425 blocks TRPV1 channels with an IC50 of 335 nM (rat) and 34 nM (human). Learn More
  7. AMG517

    Catalog No. A12727
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    TRPV1 antagonist
    AMG 517 is a potent and selective TRPV1 antagonist. Learn More
  8. Resiniferatoxin

    Catalog No. A14003
    vanilloid receptor agonist
    Resiniferatoxin is a natural analog of capsaicin (Item No. 92350) isolated from some plants of the genus Euphorbia, including E. resinifera. Learn More
  9. GSK-2193874

    Catalog No. A14201
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    TRPV4 blocker
    GSK2193874 was identified as a selective, orally active TRPV4 blocker that inhibits Ca(2+) influx through recombinant TRPV4 channels and native endothelial TRPV4 currents. Learn More
  10. GSK1016790A

    Catalog No. A15854
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    TRPV4 Activator
    GSK1016790A is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34nM in choroid plexus epithelial cells. Learn More
  11. (+)-Camphor

    Catalog No. A16423
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    Camphor is a waxy, flammable, white or transparent solid with a strong aroma, often used to relieve pain, reduce itching and treat fungal infections. It can activate TRPV1 and TRPV3 Learn More

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