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SB-705498
Catalog No. A11143 TRPV1 antagonistSB-705498 is a potent, selective and orally bioavailable TRPV1 antagonist. Learn More -
AMG517
Catalog No. A12727 TRPV1 antagonistAMG 517 is a potent and selective TRPV1 antagonist. Learn More -
A-889425
Catalog No. A13497 TRPV1 receptor antagonistA-889425 is a selective TRPV1 receptor antagonist. A-889425 blocks TRPV1 channels with an IC50 of 335 nM (rat) and 34 nM (human). Learn More -
Linoleyl ethanolamide
Catalog No. A15496 Linoleylethanolamide is an endocannabinoid that also binds to TRPV1 (Ki = 5.60 uM). Learn More -
MRS1477
Catalog No. A15498 -
Mavatrep
Catalog No. A15778 TRPV1 antagonistMavatrep is an orally bioavailable TRPV1 antagonist (Ki=6.5 nM), exhibits minimal effect on the enzymatic activity (IC50 > 25 μM) of CYP isoforms 3A4, 1A2, and 2D6. Learn More -
SB366791
Catalog No. A15857 TRPV1 receptor antagonistSB-366791 is a novel, potent, and selective, cinnamide TRPV1 antagonist. Learn More -
Capsazepine
Catalog No. A21208 TRPV1 receptorCapsazepine is a synthetic analogue of the sensory neurone excitotoxin, and an antagonist of TRPV1 receptor with an IC50 of 562 nM. Learn More -
A-1165442
Catalog No. A21516 TRPV1 antagonistA-1165442 is a potent, competitive and orally available TRPV1 antagonist with an IC50 of 9 nM for human TRPV1. Learn More -
GSK-2193874
Catalog No. A14201 TRPV4 blockerGSK2193874 was identified as a selective, orally active TRPV4 blocker that inhibits Ca(2+) influx through recombinant TRPV4 channels and native endothelial TRPV4 currents. Learn More -
Resiniferatoxin
Catalog No. A14003 vanilloid receptor agonistResiniferatoxin is a natural analog of capsaicin (Item No. 92350) isolated from some plants of the genus Euphorbia, including E. resinifera. Learn More -
GSK1016790A
Catalog No. A15854 TRPV4 ActivatorGSK1016790A is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34nM in choroid plexus epithelial cells. Learn More -
(+)-Camphor
Catalog No. A16423 Camphor is a waxy, flammable, white or transparent solid with a strong aroma, often used to relieve pain, reduce itching and treat fungal infections. It can activate TRPV1 and TRPV3 Learn More -
(Z)-Capsaicin
Catalog No. A18179 TRPV1 agonistZucapsaicin, also known as cis-Capsaicin, is a medication used to treat osteoarthritis of the knee and other neuropathic pain. It is applied three times daily for a maximum of three months. It reduces pain, and improves articular functions. Learn More -
JNJ-17203212
Catalog No. A12766 TRPV1 antagonistNJ-17203212 is a novel and selective TRPV1 antagonist, with IC50 of 65 nM and 102 nM for human TRPV1 and rat TRPV1. Learn More
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