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GM 6001

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MMP inhibitor

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Catalog No. A13320

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
GM 6001 10mg A13320-10

Regular Price: $120.00

Special Price: $108.00

GM 6001 25mg A13320-25

Regular Price: $250.00

Special Price: $225.00

GM 6001 50mg A13320-50

Regular Price: $400.00

Special Price: $360.00

GM 6001 10mM * 1mL in DMSO A13320-10mM-D

Regular Price: $106.00

Special Price: $95.40

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

GM 6001 is a potent, reversible broad spectrum inhibitor of zinc-containing proteases, including matrix metalloproteinases (MMPs).

GM 6001

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Chemical Information

Catalog Num A13320
Actions Inhibitor
M. Wt 388.5
Formula C20H28N4O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 142880-36-2
Synonyms Galardin, Ilomastat
SMILES code CC(C)C[[email protected]](CC(=O)NO)C(=O)N[[email protected]@H](CC1=CNC2=CC=CC=C21)C(=O)NC
Chemical Name (2R)-?N4-?hydroxy-?N1-?[(1S)-?1-?(1H-?indol-?3-?ylmethyl)-?2-?(methylamino)-?2-?oxoethyl]-?2-?(2-?methylpropyl)-?butanediamide

Biological Activity

Description
GM 6001 is a potent, reversible broad spectrum inhibitor of zinc-containing proteases, including matrix metalloproteinases (MMPs).
Targets
Target Value
MMP-8ki: 0.1nM
MMP-9ki: 0.2nM
MMP-26ki: 0.36nM
MMP-1ki: 0.4nM
MMP-2ki: 0.5nM
MMP-12ki: 3.6nM
MMP-7ki: 3.7nM
MMP-14ki: 13.4nM
MMP-3ki: 27nM

Solubility

Solubility (25°C)* In vitro DMSO 78 mg/mL (200.79 mM)
Water <1 mg/mL (<1 mM)
Ethanol 8 mg/mL (20.59 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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