Other inhibitors



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Catalog No. Product Name Application Product Information
A14131

NB-598

squalene epoxidase inhibitor
NB-598 is a potent competitive inhibitor of squalene epoxidase.
A14421

YL-109

-
YL-109 has ability to inhibit breast cancer cell growth and invasiveness in vitro and in vivo.
A14355

CAY10650

cPLA2α inhibitor
CAY10650 is a highly potent (IC50 = 12 nM) cPLA2α inhibitor.
A14383

Deoxynojirimycin

glucosidase I/II inhibitor
Deoxynojirimycin is a Maltase-glucoamylase (a-glucosidase I and II) inhibitor. It interferes with N-linked glycosylation.
A12981

Lesinurad

SUR inhibitor
Lesinurad is a selective uric acid re-absorption inhibitor (SURI) and is also a selective inhibitor of URAT1, a transporter in the kidney that regulates uric acid excretion from the body.
A14058

Neuropathiazol

neuronal differentiation inducer
Neuropathiazol is a synthetic small molecule that induces neuronal differentiation of adult hippocampal neural progenitor cells.
A14089

CM 346 (Afobazole)

-
CM 346 is an anxiolytic drug, produces anxiolytic and neuroprotective effects without any sedative or muscle relaxant actions.
A14329

Isomalt

-
Isomalt is a sugar substitute, a type of sugar alcohol, used primarily for its sugar-like physical properties.
A14332 SALE

JNJ-31020028

neuropeptide Y Y2 receptor antagonist
JNJ-31020028 is a novel, selective, brain-penetrant neuropeptide Y Y2 receptor antagonist
A14333

Jasmonic acid

-
Jasmonic acid is derived from the fatty acid linolenic acid.
A14347

Tazarotenic acid

-
Tazarotenic Acid is the principle active metabolite of Tazarotene.
A13839

SSR240612

bradykinin B1 receptor antagonist
SSR240612 is a new antagonist of the bradykinin B1 receptor.
A13855

AC-42

-
AC 42 is an allosteric agonist.
A13862

GW438014A

NPY Y5 receptor antagonist
GW438014A is a potent and selective neuropeptide Y Y5 receptor antagonist.
A13867

Eteplirsen (AVI-4658)

morpholino antisense oligomer
Eteplirsen is an experimental drug, currently in clinical trials.
A13870

Beloranib

METAP2 inhibitor
Beloranib, an analog of the natural chemical compound fumagillin, is an inhibitor of the enzyme METAP2.
A13875

GSK2330672

hASBT inhibitor
GSK2330672 is a highly potent, nonabsorbable apical sodium-dependent bile acid transporter inhibitor.
A13776

Ononetin

-
Ononetin is a naturally occurring deoxybenzoin.
A14406

T-5224

c-Fos inhibitor
T-5224 is a selective inhibitor of c-Fos/activator protein-1.
A14398 SALE

PFK-158

PFK-2/FBPase inhibitor
PFK-158 is an inhibitor of 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatases (PFK-2/FBPase) isoform 3 (PFKFB3) and derivative of 3-(3-pyridinyl)-1-[4-pyridinyl]-2-propen-1-one (3PO), with potential antineoplastic activity.
A14385

Afegostat

-
Afegostat was an experimental drug for the treatment of certain forms of Gaucher's disease. The substance was used in form of the tartrate. Isofagomine (IFG) is an acid ??-glucosidase (GCase) active site inhibitor that acts as a pharmacological chaperone.
A14224

Abscisic Acid

-
Abscisic Acid is a plant hormone, which is involved in many plant developmental processes, modulates ion homeostasis and metabolism.
A13309 SALE

GSK-650394

SGK1 inhibitor
GSK 650394 is a glucocorticoid- and serum-regulated kinase 1 (SGK1) inhibitor which displays antiproliferative properties against the LNCaP prostate carcinoma cell line.
A14238 SALE

Amifostine

-
Amifostine is the first approved radioprotective drug, used to decrease the risk of kidney problems caused by treatment with cisplatin.
A14241

Dicoumarol

NQO1 inhibitor
Dicoumarol is a competitive NADH quinone oxidoreductase (NQO1) inhibitor.
A12778 SALE

Lomitapide

MTP inhibitor
Lomitapide is a potent microsomal triglyceride transfer protein (MTP) inhibitor.
A14243

Phosphoramidon Disodium Salt

metalloendopeptidase inhibitor
Phosphoramidon Disodium Salt is a metalloendopeptidase inhibitor.
A14265

Meclofenoxate HCl

cholinephosphotransferase inhibitor
Meclofenoxate HCl is an anti-aging drug used to treat the symptoms of senile dementia and Alzheimer's disease, and also inhibits the activity of cholinephosphotransferase.
A14279

L-Mimosine

-
L-Mimosine is a non-protein amino acid, and acts as an iron chelator.
A14280

PTC-209 HBr

BMI-1 inhibitor

PTC-209 HBr is the hydrobromide salt of PTC-209PTC-209 is a potent and selective BMI-1 inhibitor with IC50 of 0.5 μM in HEK293T cell line, and results in irreversible reduction of cancer-initiating cells (CICs).

A14300

Home Others Others FPH1 (BRD-6125) FPH1 (BRD-6125)

-
FPH1 is a small molecule, which promotes expansion of iPS-derived hepatocytes.
A14294

MSDC-0160

mTOT-modulating insulin sensitizer
MSDC-0160 is a prototype mTOT-modulating insulin sensitizer being studied to treat diabetes and Alzheimer's disease.
A13960

SM-130686

-
SM-130686 is a potent, orally active growth hormone secretagogue, with around half the potency of the endogenous agonist ghrelin as a stimulator of growth hormone release.
A13985

DDR1-IN-1

DDR1 receptor inhibitor
DDR1-IN-1 is a potent and selective DDR1 receptor tyrosine kinase inhibitor with IC50/EC50 of 105 nM/87 nM, 4-fold less potent for DDR2 (IC50= 413 nM).
A14321

Ro 48-8071 fumarate

-
Ro 48-8071 inhibits cholesterol biosynthesis at the level of 2,3-oxidosqualene cyclase (OSC). It blocks OSC and cholesterol synthesis in HepG2 cells in the nanomolar range. A novel lipid lowering agent.
A13894

Desmethyldoxepin HCl

-
Desmethyldoxepin is the primary metabolite of doxepin, produced by metabolism at the liver. Doxepin is a tricyclic antidepressant.
A13919

Fluorocurarine chloride

sympathetic ganglioblocker
Fluorocurarine chloride is a short-acting selective sympathetic ganglioblocker with weak antagonist activity on the nicotinic receptor at the neuromuscular junction.
A14384

AB05831

beta-hexosaminidase inhibitor
AB05831 is a highly potent and specific inhibitor of beta-hexosaminidase.
A13791

Clodronate disodium

-
Clodronate disodium is the disodium salt of a nitrogen-free bisphosphonate analog of naturally occurring pyrophosphate.
A13813

Atopaxar hydrobromide

-
Atopaxar hydrobromide shows potent inhibitory effects on human platelet aggregation induced by thrombin and TRAP with IC values of 0.064 and 0.031 μM respectively.
A13824

Photochlor

-
Photochlor is a lipophilic, second-generation, chlorin-based photosensitizer. Upon intravenous administration, HPPH selectively accumulates in the cytoplasm of cancer or pre-cancerous cells.
A14014

TNP-470

MetAP-2 inhibitor
TNP 470 is an analog of Fumagillin that displays potent antiangiogenic activity in vitro. Shown to inhibit MetAP-2 (methionine aminopeptidase type II ).
A14016

Deoxygalactonojirimycin HCl

Alpha-galactosidase inhibitor
Deoxygalactonojirimycin Hydrochloride is a potent and selective Alpha-gal A (Alpha-galactosidase) inhibitor.
A13493

Ergonovine maleate

-
Ergonovine maleate is a medicine which is used in bleeding after labour and inducing or enhancing labour.
A13496

BMS-747158-02

-
BMS-747158-02 is a fluorine 18?Clabeled pyridaben derivative designed as a new myocardial perfusion imaging agent for use with positron emission tomography (PET).
A13508

N-Methyl Metribuzin

-
N-Methyl Metribuzin is an aminotriazinone and the methylamine analogue of the herbicide Metribuzin.
A13510

Methazathioprine

-
Metazathioprine is a methylated derivative of azathioprine (AZA). It demonstrated the greatest values of apparent and specific partition coefficients in n-octanol/phosphate buffer at pH 5.7 and pH 7.4 among purine derivatives such as 6-mercaptopurine (6-MP), 6-thioguanine (6-TG) and AZA.
A13512

CB-184

-
CB-184 is a useful tools for characterization of sigma 2 receptors.
A13528

Piragliatin

Glucokinase activator
Piragliatin is a novel glucokinase activator, lowers plasma glucose both in the postabsorptive state and after a glucose challenge in patients with type 2 diabetes mellitus
A13445

TH1338

-
N/A

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