Transporters



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Catalog No. Product Name Application Product Information
A13647

(-)-Blebbistcitin

myosin II inhibitor
Blebbistatin, a myosin II inhibitor, is photoinactivated by blue light.
A15785

7ACC2

MCT inhibitor
7ACC2 is a new potent MCT inhibitor with IC50 of 11 nM for inhibition of [14C]-lactate influx; new antitumor treatment targeting lactate transport in cancer cells.
A12349

Ampalex (CX-516)

-
Ampalex is an ampakine and nootropic that acts as an AMPA receptor positive allosteric modulator
A10078

Aniracetam

AMPA Receptor Inhibitor
Aniracetam is an ampakine and nootropic of the racetam chemical class purported to be considerably more potent than piracetam.
A11293

AR-C155858

MCT1 and MCT2 inhibitor
AR-C155858 is a potent inhibitor of monocarboxylate transporters MCT1 and MCT2 that binds to an intracellular site involving transmembrane helices 7-10.
A10086

Artemisinin

-
Artemisinin and its derivatives are a group of drugs that possess the most rapid action of all current drugs against Plasmodium falciparum malaria.
A14186

AZD-3965

-
AZD3965 is a selective inhibitor of monocarboxylate transporter 1 (MCT1) with a binding affinity of 1.6 nM, is 6 fold selective over MCT2 and does not inhibit MCT4 at 10 ??M.
A11961

Bafilomycin A1

ATPase inhibitor
Bafilomycin A1 prevents maturation of autophagic vacuoles by inhibiting fusion between autophagosomes and lysosomes in rat hepatoma cell line, H-4-II-E cells.
A11156

Brefeldin A

Protein translocation Inhibitor
Brefeldin A blocks binding of ADP-ribosylation factor to the Golgi apparatus and inhibits GDP-GTP exchange.
A12022

Bufalin

-
Bufalin is a cardiotonic steroid originally isolated from the Chinese toad venom.
A12024

Bufotalin

-
Bufotalin is a less potent Na+/K+-ATPase inhibitor than other bufadienolides. Potent immunosuppressor.
A11100

Canagliflozin

SGLT2 Inhibitor
Canagliflozin is an inhibitor of subtype 2 sodium-glucose transport protein (SGLT2).
A13372

CHC

MCT inhibitor
CHC is a monocarboxylic acid transport (MCT) inhibitor. Exhibits antitumoral and antiangiogenic activity in gliomas; decreases glycolytic metabolism, migration, and invasion in U251 cells.
A10213

Ciclopirox

-
Ciclopirox is currently being investigated as an alternative treatment to ketoconazole for seborrhoeic dermatitis as it suppresses growth of the yeast Malassezia furfur.It acts by inhibiting the membrane transfer system by interrupting the Na+ K+ ATPase.
A12032

Cinobufagin

-
Cinobufagin is a specific Na+/K+-ATPase inhibitor. About as active as ouabain
A10222

Citalopram Hydrobromide

-
Citalopram is a selective inhibitor of ST (5-hydroxytryptamine/serotonin transporter) and therefore is a potent and selective serotonin reuptake inhibitor.
A13321

CP 465022 hydrochloride

AMPA antagonist
CP 465022 is a selective, non-competitive AMPA antagonist with IC50 of 25 nM in rat cortical neurons that displays potent anticonvulsant activity.
A12004

Cynarin

-
Cynarin is a phenolic compound found in artichoke. It has antioxidant and choleretic properties. It is a potential immunosuppressive agent.
A10285

Dapagliflozin (BMS512148)

SGLT2 inhibitor
Dapagliflozin inhibits subtype 2 of the sodium-glucose transport proteins (SGLT2), which is responsible for at least 90% of the glucose reabsorption in the kidney.
A10319

Dipyridamole

-
Dipyridamole is a medicine that inhibits thrombus formation.
A13882

DNQX

NMDA receptor antagonist
DNQX is a non-N-methyl-D-aspartate (non-NMDA) receptor complex antagonist.
A12726

Dynasore

-
Dynasore is a non-competitive inhibitor of dynamin 1, dynamin 2 and mitochondrial dynamin (Drp1) GTPase activity
A10155

EGT1442

SGLT2 inhibitor
EGT1442 is a potent and selective SGLT2 inhibitor.
A12324

Elacridar

-
Elacridaris a prototypical BCRP inhibitor which inhibits the Bcrp1-mediated transport.
A15077

Elacridar hydrochloride

P-gp inhibitor
Elacridar hydrochloride is a P-glycoprotein inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-glycoprotein (Pgp) to investigate the role of transporters in the disposition of various test molecules.

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