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Catalog No. Product Name Application Product Information
A13647 SALE


myosin II inhibitor
Blebbistatin, a myosin II inhibitor, is photoinactivated by blue light.
A15785 SALE


MCT inhibitor
7ACC2 is a new potent MCT inhibitor with IC50 of 11 nM for inhibition of [14C]-lactate influx; new antitumor treatment targeting lactate transport in cancer cells.


A-889425 is a selective TRPV1 receptor antagonist. A-889425 blocks TRPV1 channels with an IC50 of 335 nM (rat) and 34 nM (human).
A12727 SALE


TRPV1 antagonist
AMG 517 is a potent and selective TRPV1 antagonist.
A12349 SALE

Ampalex (CX-516)

Ampalex is an ampakine and nootropic that acts as an AMPA receptor positive allosteric modulator
A10078 SALE


AMPA Receptor Inhibitor
Aniracetam is an ampakine and nootropic of the racetam chemical class purported to be considerably more potent than piracetam.


MCT1 and MCT2 inhibitor
AR-C155858 is a potent inhibitor of monocarboxylate transporters MCT1 and MCT2 that binds to an intracellular site involving transmembrane helices 7-10.
A10086 SALE


Artemisinin and its derivatives are a group of drugs that possess the most rapid action of all current drugs against Plasmodium falciparum malaria.
A14186 SALE


AZD3965 is a selective inhibitor of monocarboxylate transporter 1 (MCT1) with a binding affinity of 1.6 nM, is 6 fold selective over MCT2 and does not inhibit MCT4 at 10 ??M.

Bafilomycin A1

ATPase inhibitor
Bafilomycin A1 prevents maturation of autophagic vacuoles by inhibiting fusion between autophagosomes and lysosomes in rat hepatoma cell line, H-4-II-E cells.
A11156 SALE

Brefeldin A

Protein translocation Inhibitor
Brefeldin A blocks binding of ADP-ribosylation factor to the Golgi apparatus and inhibits GDP-GTP exchange.
A12022 SALE


Bufalin is a cardiotonic steroid originally isolated from the Chinese toad venom.


Bufotalin is a less potent Na+/K+-ATPase inhibitor than other bufadienolides. Potent immunosuppressor.
A11100 SALE


SGLT2 Inhibitor
Canagliflozin is an inhibitor of subtype 2 sodium-glucose transport protein (SGLT2).
A13372 SALE


MCT inhibitor
CHC is a monocarboxylic acid transport (MCT) inhibitor. Exhibits antitumoral and antiangiogenic activity in gliomas; decreases glycolytic metabolism, migration, and invasion in U251 cells.
A10213 SALE


Ciclopirox is currently being investigated as an alternative treatment to ketoconazole for seborrhoeic dermatitis as it suppresses growth of the yeast Malassezia furfur.It acts by inhibiting the membrane transfer system by interrupting the Na+ K+ ATPase.


Cinobufagin is a specific Na+/K+-ATPase inhibitor. About as active as ouabain
A10222 SALE

Citalopram Hydrobromide

Citalopram is a selective inhibitor of ST (5-hydroxytryptamine/serotonin transporter) and therefore is a potent and selective serotonin reuptake inhibitor.


AMPA/kainate antagonist
CNQX is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 uM for AMPA and kainate receptors, respectively, versus IC50 = 25 uM for NMDA receptors).

CNQX disodium salt

AMPA/kainate antagonist
CNQX disodium salt, water-soluble form of AMPA/kainate antagonist CNQX (GLXC-11053).

CP 465022 hydrochloride

AMPA antagonist
CP 465022 is a selective, non-competitive AMPA antagonist with IC50 of 25 nM in rat cortical neurons that displays potent anticonvulsant activity.
A12004 SALE


Cynarin is a phenolic compound found in artichoke. It has antioxidant and choleretic properties. It is a potential immunosuppressive agent.
A10285 SALE

Dapagliflozin (BMS512148)

SGLT2 inhibitor
Dapagliflozin inhibits subtype 2 of the sodium-glucose transport proteins (SGLT2), which is responsible for at least 90% of the glucose reabsorption in the kidney.


NMDA receptor antagonist
DNQX is a non-N-methyl-D-aspartate (non-NMDA) receptor complex antagonist.
A12726 SALE


Dynasore is a non-competitive inhibitor of dynamin 1, dynamin 2 and mitochondrial dynamin (Drp1) GTPase activity

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