AZD1981

Catalog No.: A13186

CRTH2 receptor antagonist

AZD1981

AZD1981 Chemical Structure

CAS NO. 802904-66-1

AZD1981, as a potent antagonist in a disease relevant cell system, inhibits DK-PGD2-induced CD11b expression in human eosinophils with IC50 of 10 nM.

Availability: In stock

Package Price Qty
5 mg
$60.00
10 mg
$100.00
25 mg
$200.00
10mM * 1mL in DMSO
$106.00
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Biological Activity

AZD1981, as a potent antagonist in a disease relevant cell system, inhibits DK-PGD2-induced CD11b expression in human eosinophils with IC50 of 10 nM.
Targets
CRTh2 (DP2) receptor
4 nM
In vitro DMSO 11 mg/mL (28.28 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.72 mL 128.58 mL 257.16 mL
0.5 mM 5.14 mL 25.72 mL 51.43 mL
1 mM 2.57 mL 12.86 mL 25.72 mL
5 mM 0.51 mL 2.57 mL 5.14 mL

*The above data is based on the productmolecular weight 388.87. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13186
Actions Antagonist
M. Wt 388.87
Formula C19H17ClN2O3S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 802904-66-1
Synonyms AZD-1981, AZD 1981
SMILES CC1=C(C2=C(N1CC(=O)O)C=CC=C2NC(=O)C)SC3=CC=C(C=C3)Cl

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