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Metabolism
Glucokinase

Glucokinase

Catalog No.

Product Name

Application

Product Information

Product Citation

A21401

Ro 28-1675

GK activator

Ro 28-1675 (Ro 0281675) is a potent allosteric GK activator with a SC1.5 value of 0.24± 0.0019 uM.

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A21562

AMG-3969

GK-GKRP disruptor

AMG-3969 is a potent glucokinase-glucokinase regulatory protein interaction (GK-GKRP) disruptor with an IC50 of 4 nM.

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A22297

Dorzagliatin

GK activator

Dorzagliatin (HMS5552), a dual-acting glucokinase (GK) activator, improves glycaemic control and pancreatic β-cell function in type 2 diabetes.

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