Biological Activity
CGP77675 is a potent Src kinase inhibitor. CGP77675 inhibited phosphorylation of peptide substrates and autophosphorylation of purified Src (IC50: 5-20 and 40 nM, respectively).
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 22.55 mL | 112.73 mL | 225.46 mL |
0.5 mM | 4.51 mL | 22.55 mL | 45.09 mL |
1 mM | 2.25 mL | 11.27 mL | 22.55 mL |
5 mM | 0.45 mL | 2.25 mL | 4.51 mL |
*The above data is based on the productmolecular weight 443.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A13821 |
---|---|
Actions | Inhibitor |
CAS No. | 234772-64-6 |
Formula | C26H29N5O2 |
M. Wt | 443.54 |
Purity | >98% |
Synonyms | CGP 77675, CGP-77675 |
SMILES | COC1=CC=CC(=C1)C2=CN(C3=C2C(=NC=N3)N)C4=CC=C(C=C4)CCN5CCC(CC5)O |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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