Amlodipine besylate (Norvasc)
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
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Discription | Amlodipine-besylate is L-type calcium channel blocker that displays antihypertensive properties. It inhibits Ca2+-induced contractions in depolarized rat aorta (IC50 = 1.9 nM) and displays vasoprotective effects in cardiovascular disease. | ||
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Catalog Num | A10069 |
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Formula | C20H25ClN2O5.C6H6O3S |
Molecular Weight | 567.1 |
CAS Number | 111470-99-6 |
SMILES | CCOC(=O)C1=C(NC(=C(C1C2=CC=CC=C2Cl)C(=O)OC)C)COCCN.C1=CC=C(C=C1)S(=O)(=O)O |
Synonyms | Istin, Norvasc |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro (25°C) | DMSO | 102 mg/mL (179.87 mM) | |
Water | Insoluble | ||
Ethanol | 13 mg/mL (22.92 mM) | ||
In vivo | 2% DMSO+30% PEG 300+2% Tween 80+ddH2O | 5 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 17.63 mL | 88.17 mL | 176.34 mL |
0.5 mM | 3.53 mL | 17.63 mL | 35.27 mL |
1 mM | 1.76 mL | 8.82 mL | 17.63 mL |
5 mM | 0.35 mL | 1.76 mL | 3.53 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2