ORY-1001 (RG-6016)
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
Not your Region? View all Distributors
Discription | ORY-1001 is an orally active and selective lysine-specific demethylase LSD1/KDM1A inhibitor with IC50 of <20 nM, with high selectivity against related FAD dependent aminoxidases. Phase 1. | ||
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Catalog Num | A15893 |
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Formula | C15H22N2.2HCl |
Molecular Weight | 303.27 |
CAS Number | 1431326-61-2 |
SMILES | NC1CCC(N[C@@H]2C[C@H]2C3=CC=CC=C3)CC1.Cl.Cl |
Synonyms | RG6016, RG-6016 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 4 mg/mL (13.18 mM) | |
Water | 53 mg/mL (174.76 mM) | ||
Ethanol | Warmed: 3 mg/mL (9.89 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 32.97 mL | 164.87 mL | 329.74 mL |
0.5 mM | 6.59 mL | 32.97 mL | 65.95 mL |
1 mM | 3.3 mL | 16.49 mL | 32.97 mL |
5 mM | 0.66 mL | 3.3 mL | 6.59 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2