Tegaserod maleate
5-HT antagonist
Important Notice: For research use only. We do not sell to patients.
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5-HT antagonist
Important Notice: For research use only. We do not sell to patients.
Not your Region? View all Distributors
Discription | Tegaserod functions as a motility stimulant, achieving its desired therapeutic effects through activation of the 5-HT4 receptors of the enteric nervous system in the gastrointestinal tract. It also stimulates gastrointestinal motility and the peristaltic reflex, and allegedly reduces abdominal pain. Additionally, tegaserod is a 5-HT2B receptor antagonist. | ||
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Catalog Num | A11743 |
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Formula | C16H23N5O.C4H4O4 |
Molecular Weight | 417.46 |
CAS Number | 189188-57-6 |
SMILES | CCCCCN=C(N)NN/C=C/1\C=NC2=C1C=C(C=C2)OC.C(=C\C(=O)O)\C(=O)O |
Synonyms | Zelnorm |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 72 mg/mL (172.47 mM) | |
Water | Insoluble | ||
Ethanol | 7 mg/mL (16.77 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 23.95 mL | 119.77 mL | 239.54 mL |
0.5 mM | 4.79 mL | 23.95 mL | 47.91 mL |
1 mM | 2.4 mL | 11.98 mL | 23.95 mL |
5 mM | 0.48 mL | 2.4 mL | 4.79 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2