GS-9973 (Entospletinib)
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
Not your Region? View all Distributors
Discription | GS-9973 is an oral inhibitor of spleen tyrosine kinase (Syk), with potential antineoplastic activity. | ||
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Targets |
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Catalog Num | A13884 |
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Formula | C23H21N7O |
Molecular Weight | 411.46 |
CAS Number | 1229208-44-9 |
SMILES | C1COCCN1C2=CC=C(C=C2)NC3=NC(=CN4C3=NC=C4)C5=CC6=C(C=C5)C=NN6 |
Synonyms | GS9973, GS 9973, Entospletinib |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro (25°C) | DMSO | Warmed: 26 mg/mL (63.18 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
In vivo | 4% DMSO+30% PEG 300+5% Tween 80+ddH2O | 2.3 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 24.3 mL | 121.52 mL | 243.04 mL |
0.5 mM | 4.86 mL | 24.3 mL | 48.61 mL |
1 mM | 2.43 mL | 12.15 mL | 24.3 mL |
5 mM | 0.49 mL | 2.43 mL | 4.86 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2