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GDC-0032 is a potent, next-generation PI3 inhibitor targeting PI3 alpha.
Targets
| Target | Value |
|---|---|
| PI3Kδ | ki: 0.12nM |
| PI3Kα | ki: 0.29nM |
| PI3Kγ | ki: 0.97nM |
| PI3Kβ | ki: 9.1nM |
| C2β | IC50: 292nM |
| hVps34 | IC50: 374nM |
| mTOR | ki: 1.2μM |
| DNA-PK | IC50: >4.8μM |
| C2α | IC50: >10μM |
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 21.71 mL | 108.57 mL | 217.14 mL |
| 0.5 mM | 4.34 mL | 21.71 mL | 43.43 mL |
| 1 mM | 2.17 mL | 10.86 mL | 21.71 mL |
| 5 mM | 0.43 mL | 2.17 mL | 4.34 mL |
*The above data is based on the productmolecular weight 460.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Chemical Properties
| Catalog Num | A12831 |
|---|---|
| Actions | Inhibitor |
| M. Wt | 460.53 |
| Formula | C24H28N8O2 |
| Solubility | DMSO |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 1282512-48-4 |
| Synonyms | GDC 0032, GDC0032 |
| SMILES | CC1=NN(C(=N1)C2=CN3CCOC4=C(C3=N2)C=CC(=C4)C5=CN(N=C5)C(C)(C)C(=O)N)C(C)C |
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