GDC-0032 (Taselisib)

Catalog No.: A12831

PI3K inhibitor

GDC-0032 (Taselisib)

GDC-0032 (Taselisib) Chemical Structure

CAS NO. 1282512-48-4

GDC-0032 is a potent, next-generation PI3 inhibitor targeting PI3 alpha.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $70.00

Special Price $63.00

10 mg

Regular Price: $110.00

Special Price $99.00

25 mg

Regular Price: $200.00

Special Price $180.00

50 mg

Regular Price: $290.00

Special Price $261.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

GDC-0032 is a potent, next-generation PI3 inhibitor targeting PI3 alpha.
Targets
Target Value
PI3Kδki: 0.12nM
PI3Kαki: 0.29nM
PI3Kγki: 0.97nM
PI3Kβki: 9.1nM
C2βIC50: 292nM
hVps34IC50: 374nM
mTORki: 1.2μM
DNA-PKIC50: >4.8μM
C2αIC50: >10μM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.71 mL 108.57 mL 217.14 mL
0.5 mM 4.34 mL 21.71 mL 43.43 mL
1 mM 2.17 mL 10.86 mL 21.71 mL
5 mM 0.43 mL 2.17 mL 4.34 mL

*The above data is based on the productmolecular weight 460.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A12831
Actions Inhibitor
M. Wt 460.53
Formula C24H28N8O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1282512-48-4
Synonyms GDC 0032, GDC0032
SMILES CC1=NN(C(=N1)C2=CN3CCOC4=C(C3=N2)C=CC(=C4)C5=CN(N=C5)C(C)(C)C(=O)N)C(C)C

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