Catalog No.: A14433
NOX1/4 inhibitor
GKT137831 is a first in class inhibitor targeting NOX1 and NOX4 enzymes.
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GKT137831 5mg
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GKT137831 10mg
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GKT137831 25mg
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GKT137831 10mM * 1mL in DMSO
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Adooq Products cited in reputable paper
Adooq's GKT137831 has been cited by 1 publications
  • Chia-Hui Huang, .et al. , Toxicol Appl Pharmacol, 2020, Apr 17;397:115013 PMID: 32305283
  • Biological Activity
    Discription GKT137831 is a first in class inhibitor targeting NOX1 and NOX4 enzymes.
    Target Value
    Product Information
    Catalog Num A14433
    Formula C21H19ClN4O2
    Molecular Weight 394.85
    CAS Number 1218942-37-0
    SMILES CN1C(=O)C=C2C(=C1C3=CC(=CC=C3)N(C)C)C(=O)N(N2)C4=CC=CC=C4Cl
    Synonyms GKT-137831, GKT 137831

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

    In vitro (25°C) DMSO Warmed: 72 mg/mL (182.34 mM)
    Water Insoluble
    Ethanol Insoluble
    In vivo 2% DMSO+2% Tween 80+30% PEG 300+ddH2O 8 mg/mL
    * <1 mg/ml means slightly soluble or insoluble.
    * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
    Preparing Stock Solutions
    Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
    0.1 mM 25.33 mL 126.63 mL 253.26 mL
    0.5 mM 5.07 mL 25.33 mL 50.65 mL
    1 mM 2.53 mL 12.66 mL 25.33 mL
    5 mM 0.51 mL 2.53 mL 5.07 mL
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    Calculate the dilution required to prepare a stock solution.
    This equation is commonly abbreviated as: C1V1 = C2V2

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