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MLN 2480 is an oral, selective pan-Raf kinase inhibitor in chinical trials.
Targets
| Raf | ||||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 19.75 mL | 98.76 mL | 197.52 mL |
| 0.5 mM | 3.95 mL | 19.75 mL | 39.5 mL |
| 1 mM | 1.98 mL | 9.88 mL | 19.75 mL |
| 5 mM | 0.4 mL | 1.98 mL | 3.95 mL |
*The above data is based on the productmolecular weight 506.29. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A11240 |
|---|---|
| Actions | Inhibitor |
| M. Wt | 506.29 |
| Formula | C17H12Cl2F3N7O2S |
| Solubility | DMSO |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 1096708-71-2 |
| Synonyms | MLN-2480,BIIB 024, BIIB-024 |
| SMILES | C[[email protected]](C1=NC=C(S1)C(=O)NC2=NC=C(C(=C2)C(F)(F)F)Cl)NC(=O)C3=C(C(=NC=N3)N)Cl |
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