Nalfurafine hydrochloride

Catalog No.: A12579

opioid κ-selective agonist

Nalfurafine hydrochloride

Nalfurafine hydrochloride Chemical Structure

CAS NO. 152658-17-8

Nalfurafine hydrochloride is a kappa-opioid receptor agonist

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  • Dunn AD, .et al. Signaling Properties of Structurally Diverse Kappa Opioid Receptor Ligands: Toward in Vitro Models of in Vivo Responses, ACS Chem Neurosci, 2019, Aug 21;10(8):3590-3600 PMID: 31313902
  • Anika Mann, .et al. Agonist-selective NOP receptor phosphorylation correlates in vitro and in vivo and reveals differential post-activation signaling by chemically diverse agonists, Sci Signal, 2019, Mar 26;12(574). pii: eaau8072 PMID: 30914485
  • Snyder LM, .et al. Kappa Opioid Receptor Distribution and Function in Primary Afferents, Neuron, 2018, Sep 19;99(6):1274-1288.e6 PMID: 30236284

Biological Activity

Nalfurafine hydrochloride is a kappa-opioid receptor agonist
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.49 mL 97.46 mL 194.92 mL
0.5 mM 3.9 mL 19.49 mL 38.98 mL
1 mM 1.95 mL 9.75 mL 19.49 mL
5 mM 0.39 mL 1.95 mL 3.9 mL

*The above data is based on the productmolecular weight 513.03. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12579
Actions Agonist
M. Wt 513.03
Formula C28H33ClN2O5
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 152658-17-8
Synonyms AC-820, TRK-820, Remitch
SMILES CN([[email protected]@H]1CC[[email protected]]2([[email protected]]3CC4=C5[[email protected]]2([[email protected]]1OC5=C(C=C4)O)CCN3CC6CC6)O)C(=O)/C=C/C7=COC=C7.Cl

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