GABA Receptors

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  1. GABA antagonist

    Cloflubicyne is a potent non-competitive GABA antagonist, convulsant, laboratory insecticide.
  2. DSP-0565 is a strong, broad-spectrum anti-epileptic drug (AED) candidate with unique GABAergic function.
  3. Lotilaner is an insecticide (veterinary drug).
  4. GABAA α5 modulator

    ONO-8590580 is a GABAA α5 negative allosteric modulator.
  5. GABAB receptor agonist

    rac-BHFF is a selective GABAB receptor agonist.

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