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Publications citing Adooq Products
Chemical Information
| Catalog Num | A15196 |
|---|---|
| Actions | Inhibitor |
| M. Wt | 460.33 |
| Formula | C17H19Cl2N5O4S |
| Solubility | DMSO |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 902156-99-4 |
| Synonyms | LCQ-195, AT-9311, NVP LCQ195, LCQ 195, AT9311, AT 9311 |
| SMILES code | CS(=O)(=O)N1CCC(CC1)NC(=O)C2=C(C=NN2)NC(=O)C3=C(C=CC=C3Cl)Cl |
| Chemical Name | 4-[(2,6-dichlorobenzoyl)amino]-N-(1-methylsulfonylpiperidin-4-yl)-1H-pyrazole-5-carboxamide |
Description |
NVP-LCQ195 is a small molecule heterocyclic inhibitor of CDK1, CDK2, CDK3 and CDK5 with IC50 of 1-42 nM. | |||||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 21.72 mL | 108.62 mL | 217.24mL |
| 0.5 mM | 4.34 mL | 21.72 mL | 43.45 mL |
| 1 mM | 2.17 mL | 10.86 mL | 21.72 mL |
| 5 mM | 0.43 mL | 2.17 mL | 4.34 mL |
*The above data is based on the productmolecular weight 460.33. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
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