Others

(±)-WS75624B is an endothelin converting enzyme (ECE) inhibitor with an IC50 of 0.03 μg/mL.

Sotirimod is an immunostimulant, and can potentially treat for actinic keratosis.

Anti-Heart Failure Agent 1 an orally available compound suitable for the treatment of heart failure without inducing nausea, vomiting and restlessness.

CGS 15435, a potent thromboxane (TxA2) synthetase inhibitor with an IC50 of 1 nM, has a selectivity for Tx synthetase 100000-fold greater than that for cyclooxygenase, PGI2 synthetase and lipoxygenase enzymes.

Chymase-IN-1 is a potent, selective, orally active, nonpeptide inhibitor of human mast cell chymase with an IC50 of 29 nM.

Cinperene is an atropine-like drug which can block pilocarpine-induced lacrimation and salivation.

Nafocare B1 is a synthetic immune biological response modifier.

F 16915 is a docosahexaenoic acid derivative which can prevent heart failure-induced atrial fibrillation.

SC-52012 is an orally active fibrinogen receptor antagonist, with antiplatelet activities.

FR194738 is a squalene epoxidase inhibitor. FR194738 inhibits squalene epoxidase activity in HepG2 cell homogenates with an IC50 of 9.8 nM.

RO5203648 hydrochloride is a partial agonist of Trace amine-associated receptor 1 (TAAR1).