Reboxetine mesylate

Catalog No.: A11919

Reboxetine mesylate

Reboxetine mesylate Chemical Structure

CAS NO. 98769-84-7

Reboxetine is an antidepressant compound that selectively inhibits norepinephrine uptake (IC50s = 8.2 and 1,070 nM for norepinephrine and serotonin transporters, respectively). It displays greater than 1,000-fold affinity for binding rat norepinephrine receptors compared to serotonin, histamine, acetylcholine, or dopamine receptors (Kis = 1.1, 129, 1,400, 3,900, and >10,000 nM, respectively).

Availability: In stock

Package Price Qty
5 mg

Regular Price: $40.00

Special Price $32.00

10 mg

Regular Price: $70.00

Special Price $56.00

25 mg

Regular Price: $120.00

Special Price $96.00

50 mg

Regular Price: $200.00

Special Price $160.00

10mM * 1mL in DMSO

Regular Price: $92.00

Special Price $73.60

Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Reboxetine is an antidepressant compound that selectively inhibits norepinephrine uptake (IC50s = 8.2 and 1,070 nM for norepinephrine and serotonin transporters, respectively). It displays greater than 1,000-fold affinity for binding rat norepinephrine receptors compared to serotonin, histamine, acetylcholine, or dopamine receptors (Kis = 1.1, 129, 1,400, 3,900, and >10,000 nM, respectively).
Targets
norepinephrine reuptake
8.2 nM(Ki)
In vitro DMSO 81 mg/mL (197.8 mM)
Water 81 mg/mL (197.8 mM)
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.42 mL 122.1 mL 244.2 mL
0.5 mM 4.88 mL 24.42 mL 48.84 mL
1 mM 2.44 mL 12.21 mL 24.42 mL
5 mM 0.49 mL 2.44 mL 4.88 mL

*The above data is based on the productmolecular weight 409.5. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11919
CAS No. 98769-84-7
Formula C19H23NO3.CH4SO3
M. Wt 409.5
Purity >98%
SMILES CCOC1=CC=CC=C1O[[email protected]@H]([[email protected]]2CNCCO2)C3=CC=CC=C3.CS(=O)(=O)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy Reboxetine mesylate | Reboxetine mesylate Supplier | purchase | cost | manufacturer | order | distributor | buy 98769-84-7| 98769-84-7 Supplier | purchase 98769-84-7 | 98769-84-7 cost | 98769-84-7 manufacturer | order 98769-84-7 | 98769-84-7 distributor
Rewards