Total item
Cart Subtotal
$0.00 Biological Activity
RKI-1447 is a potent inhibitor of the Rho-associated ROCK kinases with anti-invasive and antitumor activities in breast cancer.
Targets
| ROCK2 | ROCK1 | |||
| 6.2 nM | 14.5 nM |
| In vitro (25°C) | DMSO | 65 mg/mL (199.16 mM) | |
| Water | <1 mg/mL (<1 mM) | ||
| Ethanol | <1 mg/mL (<1 mM) | ||
| In vivo | 15% Captisol | 30 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 30.64 mL | 153.2 mL | 306.4 mL |
| 0.5 mM | 6.13 mL | 30.64 mL | 61.28 mL |
| 1 mM | 3.06 mL | 15.32 mL | 30.64 mL |
| 5 mM | 0.61 mL | 3.06 mL | 6.13 mL |
*The above data is based on the productmolecular weight 326.37. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A13067 |
|---|---|
| Actions | Inhibitor |
| M. Wt | 326.37 |
| Formula | C16H14N4O2S |
| Solubility | DMSO |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 1342278-01-6 |
| Synonyms | RKI1447; RKI 1447. ROCK Inhibitor XIII |
| SMILES | C1=CC(=CC(=C1)O)CNC(=O)NC2=NC(=CS2)C3=CC=NC=C3 |
Product Tags
Product Questions
Product Questions
No Questions
Keywords:buy RKI-1447 | RKI-1447 Supplier | purchase | cost | manufacturer | order | distributor | buy 1342278-01-6| 1342278-01-6 Supplier | purchase 1342278-01-6 | 1342278-01-6 cost | 1342278-01-6 manufacturer | order 1342278-01-6 | 1342278-01-6 distributor
Contact information
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: [email protected]
Not your Region? View all Distributors
Adooq Quality Guarantee
We promise all products perform as described.