Talnetant hydrochloride

Catalog No.: A15255

NK3 receptor antagonist

Talnetant hydrochloride

Talnetant hydrochloride Chemical Structure

CAS NO. 204519-66-4

Talnetant Hcl is a potent and selective NK3 receptor antagonist(ki=1.4 nM, hNK-3-CHO); 100-fold selective for the hNK-3 versus hNK-2 receptor, with no affinity for the hNK-1 at concentrations up to 100 uM.

Availability: In stock

Package Price Qty
10 mg
$128.00
25 mg
$280.00
50 mg
$500.00
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Biological Activity

Talnetant Hcl is a potent and selective NK3 receptor antagonist(ki=1.4 nM, hNK-3-CHO); 100-fold selective for the hNK-3 versus hNK-2 receptor, with no affinity for the hNK-1 at concentrations up to 100 uM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.87 mL 119.35 mL 238.71 mL
0.5 mM 4.77 mL 23.87 mL 47.74 mL
1 mM 2.39 mL 11.94 mL 23.87 mL
5 mM 0.48 mL 2.39 mL 4.77 mL

*The above data is based on the productmolecular weight 418.92. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15255
Actions Antagonist
CAS No. 204519-66-4
Formula C25H23ClN2O2
M. Wt 418.92
Purity >98%
Synonyms SB-223412 hydrochloride, SB223412 hydrochloride, SB 223412 hydrochloride, SB 223412-A
SMILES CCC(C1=CC=CC=C1)NC(=O)C2=C(C(=NC3=CC=CC=C32)C4=CC=CC=C4)O.Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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