Tegaserod maleate

Catalog No.: A11743

Tegaserod maleate

Tegaserod maleate Chemical Structure

CAS NO. 189188-57-6

Tegaserod functions as a motility stimulant, achieving its desired therapeutic effects through activation of the 5-HT4 receptors of the enteric nervous system in the gastrointestinal tract. It also stimulates gastrointestinal motility and the peristaltic reflex, and allegedly reduces abdominal pain. Additionally, tegaserod is a 5-HT2B receptor antagonist.

Availability: In stock

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10 mg

Regular Price: $90.00

Special Price $72.00

50 mg

Regular Price: $280.00

Special Price $224.00

100 mg

Regular Price: $480.00

Special Price $384.00

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Biological Activity

Tegaserod functions as a motility stimulant, achieving its desired therapeutic effects through activation of the 5-HT4 receptors of the enteric nervous system in the gastrointestinal tract. It also stimulates gastrointestinal motility and the peristaltic reflex, and allegedly reduces abdominal pain. Additionally, tegaserod is a 5-HT2B receptor antagonist.
In vitro DMSO 72 mg/mL (172.47 mM)
Water Insoluble
Ethanol 7 mg/mL (16.77 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.95 mL 119.77 mL 239.54 mL
0.5 mM 4.79 mL 23.95 mL 47.91 mL
1 mM 2.4 mL 11.98 mL 23.95 mL
5 mM 0.48 mL 2.4 mL 4.79 mL

*The above data is based on the productmolecular weight 417.46. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11743
CAS No. 189188-57-6
Formula C16H23N5O.C4H4O4
M. Wt 417.46
Purity >98%
Synonyms Zelnorm
SMILES CCCCCN=C(N)NN/C=C/1\C=NC2=C1C=C(C=C2)OC.C(=C\C(=O)O)\C(=O)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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