Telatinib (BAY 57-9352)

Catalog No.: A10903

VEGFR-2 inhibitor

Telatinib (BAY 57-9352) Chemical Structure

CAS NO. 332012-40-5

Telatinib (BAY 57-9352) is an orally available, small-molecule inhibitor of vascular endothelial growth factor receptors 2 and 3 (VEGFR-2/-3) and platelet-derived growth factor receptor β tyrosine kinases.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $90.00

Special Price $72.00

10 mg

Regular Price: $160.00

Special Price $128.00

50 mg

Regular Price: $450.00

Special Price $360.00

100 mg

Regular Price: $750.00

Special Price $600.00

10mM * 1mL in DMSO
$133.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Telatinib (BAY 57-9352) is an orally available, small-molecule inhibitor of vascular endothelial growth factor receptors 2 and 3 (VEGFR-2/-3) and platelet-derived growth factor receptor β tyrosine kinases.
Targets
c-Kit VEGFR3 VEGFR2 PDGFRα
1 nM4 nM6 nM15 nM
In vitro DMSO 82 mg/mL (200.08 mM)
Water <1 mg/mL (<1 mM)
Ethanol 1 mg/mL (2.44 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.4 mL 122.01 mL 244.02 mL
0.5 mM 4.88 mL 24.4 mL 48.8 mL
1 mM 2.44 mL 12.2 mL 24.4 mL
5 mM 0.49 mL 2.44 mL 4.88 mL

*The above data is based on the productmolecular weight 409.8 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10903
Actions Inhibitor
M. Wt 409.8
Formula C20H16ClN5O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 332012-40-5
Synonyms BAY57-9352
SMILES CNC(=O)C1=NC=CC(=C1)COC2=NN=C(C3=C2OC=C3)NC4=CC=C(C=C4)Cl

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