Biological Activity
TGR5 Receptor Agonist is a potent TGR5(GPCR19) agonist, showed improved potency in the U2-OS cell assay (pEC50 = 6.8) and in melanophore cells (pEC50 = 7.5).
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 27.68 mL | 138.42 mL | 276.84 mL |
0.5 mM | 5.54 mL | 27.68 mL | 55.37 mL |
1 mM | 2.77 mL | 13.84 mL | 27.68 mL |
5 mM | 0.55 mL | 2.77 mL | 5.54 mL |
*The above data is based on the productmolecular weight 361.22. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A13732 |
---|---|
Actions | Agonist |
M. Wt | 361.22 |
Formula | C18H14Cl2N2O2 |
Solubility | DMSO |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 1197300-24-5 |
SMILES | CC1=C(C(=NO1)C2=CC=CC=C2Cl)C(=O)N(C)C3=CC=C(C=C3)Cl |
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