Adenosine Receptors

CGS 15943 is a potent, non-selective Adenosine A Receptor antagonist. It is orally active in vivo.

MRE3008F20 is a highly potent and selective antagonist of adenosine A3 receptor (AA3R), inhibits agonist-induced cAMP elevation in resting T lymphocytes with an IC50 of 5 nM.