JavaScript seems to be disabled in your browser. For the best experience on our site, be sure to turn on Javascript in your browser.

Home
GPCR/G Protein
Calcium-Sensing Receptor

Calcium-Sensing Receptor

Catalog No.

Product Name

Application

Product Information

Product Citation

A19779

GSK3004774

CaSR agonist

GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR, respectively. GSK3004774 shows an EC50 of 50 nM for human CaSR.

Quick View
A21169

SB-423557

Calcium-sensing receptor (CaR) antagonist

SB-423557 is an orally active calcium-sensing receptor (CaR) antagonist (IC50=520 nM), precursor of SB-423562 (IC50=73 nM).

Quick View