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GPCR/G Protein
Opioid Receptors

Opioid Receptors

Catalog No.

Product Name

Application

Product Information

Product Citation

A15149

LY2795050

k-opioid receptor antagonist

LY2795050 is a novel selective κ-opioid Receptor (KOR) antagonist (IC50=0.72 nM) and has the potential as a PET tracer to image KOR in vivo.

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A16902

SR-17018

MOR agonist

SR17018 is an mu-opioid-receptor (MOR) agonist with an EC50 of 97 nM.

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- Rob Hill, .et al. , Br J Pharmacol, 2023, Jul 24 PMID: 37489013
A22124

BMS-986188

δ-opioid receptor modulator

BMS-986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.

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A22125

BMS-986187

δ-opioid receptor modulator

BMS-986187 is a potent and selective positive allosteric modulator (PAM) of the δ-opioid receptor and a G-protein-biased allosteric agonist.

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