AR-C155858

Catalog No.: A11293

MCT1 and MCT2 inhibitor

AR-C155858 Chemical Structure

CAS NO. 496791-37-8

AR-C155858 is a potent inhibitor of monocarboxylate transporters MCT1 and MCT2 that binds to an intracellular site involving transmembrane helices 7-10.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $360.00

Special Price $288.00

10 mg

Regular Price: $600.00

Special Price $480.00

25 mg

Regular Price: $1,200.00

Special Price $960.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

AR-C155858 is a potent inhibitor of monocarboxylate transporters MCT1 and MCT2 that binds to an intracellular site involving transmembrane helices 7-10.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.67 mL 108.34 mL 216.68 mL
0.5 mM 4.33 mL 21.67 mL 43.34 mL
1 mM 2.17 mL 10.83 mL 21.67 mL
5 mM 0.43 mL 2.17 mL 4.33 mL

*The above data is based on the productmolecular weight 461.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11293
Actions Inhibitor
M. Wt 461.5
Formula C21H27N5O5S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 496791-37-8
Synonyms AR-C 155858
SMILES CC1=C(C(=NN1)C)CC2=C(C3=C(S2)N(C(=O)N(C3=O)C)CC(C)C)C(=O)N4C[[email protected]@H](CO4)O
1. Ovens et al (2010) The inhibition of monocarboxylate transporter 2 (MCT2) by AR-C155858 is modulated by the associated ancillary protein. Biochem.J. 431 217. PMID: 20695846.
2.Ovens et al (2010) AR-C155858 is a potent inhibitor of monocarboxylate transporters MCT1 and MCT2 that binds to an intracellular site involving transmembrane helices 7-10. Biochem.J. 425 523. PMID: 19929853.

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