GABA Receptors

Lorediplon is a novel non-benzodiazepine, hypnotic drug acting as a GABAA receptor modulator,

CTP354 a novel deuterated subtype-selective GABA(A) modulator.

Loreclezole, an antiepileptic compound, is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit containing receptors.