PHA-767491

Catalog No.: A11164

Cdc7/cdk9 inhibitor

PHA-767491

PHA-767491 Chemical Structure

CAS NO. 845714-00-3

PHA-767491 is a potent, ATP-competitive dual cdc7/cdk9 inhibitor (IC50 values are 10 and 34 nM respectively) that prevents initiation of DNA replication.

Availability: In stock

Package Price Qty
10 mg
$70.00
50 mg
$280.00
100 mg
$490.00
10mM * 1mL in DMSO
$76.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Qi Li, .et al. CDC7-dependent transcriptional regulation of RAD54L is essential for tumorigenicity and radio-resistance of glioblastoma, Transl Oncol, 2018, Apr; 11(2): 300-306 PMID: 29413763

Biological Activity

PHA-767491 is a potent, ATP-competitive dual cdc7/cdk9 inhibitor (IC50 values are 10 and 34 nM respectively) that prevents initiation of DNA replication.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 46.9 mL 234.48 mL 468.96 mL
0.5 mM 9.38 mL 46.9 mL 93.79 mL
1 mM 4.69 mL 23.45 mL 46.9 mL
5 mM 0.94 mL 4.69 mL 9.38 mL

*The above data is based on the productmolecular weight 213.24. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11164
Actions Inhibitor
CAS No. 845714-00-3
Formula C12H11N3O
M. Wt 213.24
Purity >98%
Synonyms PHA767491
SMILES C1CNC(=O)C2=C1NC(=C2)C3=CC=NC=C3
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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