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GPCR/G Protein
Adenosine Receptors

Adenosine Receptors

Catalog No.

Product Name

Application

Product Information

Product Citation

A12880

ST3932

Adenosine A2A receptor antagonist

ST3932 is a metabolite of ST1535, acts as an antagonist of adenosine A2A receptor, with Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively.

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A16870

MRS1186

Adenosine A3 receptor antagonist

MRS1186 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 7.66 nM.

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A16871

MRS1177

Adenosine A3 receptor antagonist

MRS1177 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 0.3 nM.

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A20116

BAY-545

A2B adenosine receptor antagonist

BAY-545 is a potent and selective A2B adenosine receptor antagonist, with an IC50 of 59 nM.

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A21649

Rolofylline

adenosine A1 receptor antagonist

Rolofylline (KW-3902) is a potent, selective adenosine A1 receptor antagonist that is under development for the treatment of patients with acute congestive heart failure and renal impairment.

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A21990

Derenofylline

adenosine A1 receptor antagonist

Derenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively.

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