ARRY-543 (Varlitinib, ASLAN001)

Catalog No.: A12868

ErbB inhibitor

ARRY-543 (Varlitinib, ASLAN001)

ARRY-543 (Varlitinib, ASLAN001) Chemical Structure

CAS NO. 114629-86-8

ARRY-543 is a novel, oral ErbB family inhibitor that, unlike approved ErbB inhibitors, targets all members of the ErbB family, including ErbB3, either directly or indirectly, and has potential advantages in treating tumors that signal through multiple ErbB family members.

Availability: In stock

Package Price Qty
5 mg
$350.00
10 mg
$650.00
25 mg
$1,200.00
50 mg
$2,000.00
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Biological Activity

ARRY-543 is a novel, oral ErbB family inhibitor that, unlike approved ErbB inhibitors, targets all members of the ErbB family, including ErbB3, either directly or indirectly, and has potential advantages in treating tumors that signal through multiple ErbB family members.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 12.85 mL 64.25 mL 128.51 mL
0.5 mM 2.57 mL 12.85 mL 25.7 mL
1 mM 1.29 mL 6.43 mL 12.85 mL
5 mM 0.26 mL 1.29 mL 2.57 mL

*The above data is based on the productmolecular weight 778.15. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12868
Actions Inhibitor
CAS No. 114629-86-8
Formula C36H35ClN6O6S3
M. Wt 778.15
Purity >98%
Synonyms ARRY543,ARRY 543
SMILES ClC1=CC(NC2=NC=NC3=CC=C(NC4=N[[email protected]](C)CO4)C=C32)=CC=C1OCC5=NC=CS5.CC6=CC=C(S(O)=O)C=C6.CC7=CC=C(S(O)=O)C=C7
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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