Imidazoline Receptor
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Moxonidine Hydrochloride
Catalog No. A13416 imidazoline receptor 1 agonistMoxonidine hydrochloride is a centrally acting antihypertensive agent. Learn More -
Moxonidine HCl
Catalog No. A11741 imidazoline receptor 1 agonistMoxonidine is a selective agonist at the imidazoline receptor subtype 1 (I1). Moxonidine causes a decrease in sympathetic nervous system activity and, therefore, a decrease in blood pressure. Learn More -
Clonidine hydrochloride
Catalog No. A10232 Alpha adrenergic agonistClonidine is classified as a centrally acting alpha adrenergic agonist.Clonidine acts centrally as an imidazoline receptor agonist. Learn More -
Rilmenidine
Catalog No. A10794 α2 adrenergic agonistRilmenidine is a second-generation imidazoline-α2 adrenergic agonist. Learn More -
Rilmenidine Phosphate
Catalog No. A14256 I(1) imidazoline receptor agonistRilmenidine Phosphate is a selective I(1) imidazoline receptor agonist. Learn More -
Guanabenz acetate
Catalog No. A13635 2A-AR adrenergic agonistGuanabenz acetate is an a2A-AR adrenergic agonist and IGRS (imidazoline I2 binding site) selective ligand. Learn More -
KU14R
Catalog No. A13987 I3 receptor AntagonistKU14R is an antagonist of the pancreatic β-cell atypical imidazoline binding site (putative I3 receptor). KU14R has also been shown to selectively block efaroxan-induced insulin secretion. Learn More -
Idazoxan Hydrochloride
Catalog No. A13409 α2- adrenoceptor antagonist / I2 imidazoline receptor agonistIdazoxan hydrochloride is an α2-AR adrenoceptor antagonist and potential I2 imidazoline receptor agonist. Also displays I1 imidazoline receptor antagonist activity. (pKi values are 5.90, 7.22, 8.01, 7.43, and 7.7 for I1, I2, α 2A, α2B, and α 2C receptors respectively). Learn More