Imidazoline Receptor

8 Item(s)

per page

Set Descending Direction
  1. Moxonidine Hydrochloride

    Catalog No. A13416
    Quick View
    imidazoline receptor 1 agonist
    Moxonidine hydrochloride is a centrally acting antihypertensive agent. Learn More
  2. Moxonidine HCl

    Catalog No. A11741
    Quick View
    imidazoline receptor 1 agonist
    Moxonidine is a selective agonist at the imidazoline receptor subtype 1 (I1). Moxonidine causes a decrease in sympathetic nervous system activity and, therefore, a decrease in blood pressure. Learn More
  3. Clonidine hydrochloride

    Catalog No. A10232
    Quick View
    Alpha adrenergic agonist
    Clonidine is classified as a centrally acting alpha adrenergic agonist.Clonidine acts centrally as an imidazoline receptor agonist. Learn More
  4. Rilmenidine

    Catalog No. A10794
    Quick View
    α2 adrenergic agonist
    Rilmenidine is a second-generation imidazoline-α2 adrenergic agonist. Learn More
  5. Rilmenidine Phosphate

    Catalog No. A14256
    Quick View
    I(1) imidazoline receptor agonist
    Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist. Learn More
  6. Guanabenz acetate

    Catalog No. A13635
    Quick View
    2A-AR adrenergic agonist
    Guanabenz acetate is an a2A-AR adrenergic agonist and IGRS (imidazoline I2 binding site) selective ligand. Learn More
  7. KU14R

    Catalog No. A13987
    Quick View
    I3 receptor Antagonist
    KU14R is an antagonist of the pancreatic β-cell atypical imidazoline binding site (putative I3 receptor). KU14R has also been shown to selectively block efaroxan-induced insulin secretion. Learn More
  8. Idazoxan Hydrochloride

    Catalog No. A13409
    Quick View
    α2- adrenoceptor antagonist / I2 imidazoline receptor agonist
    Idazoxan hydrochloride is an α2-AR adrenoceptor antagonist and potential I2 imidazoline receptor agonist. Also displays I1 imidazoline receptor antagonist activity. (pKi values are 5.90, 7.22, 8.01, 7.43, and 7.7 for I1, I2, α 2A, α2B, and α 2C receptors respectively). Learn More

8 Item(s)

per page

Set Descending Direction
Rewards