Neurotensin Receptors
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SR 48692
Catalog No. A11770 NT AntagonistSR 48692 represents a new, potent, nonpeptide antagonist radioligand of the NT receptor that differentiates between agonist- and antagonist-receptor interactions. Learn More -
ML314
Catalog No. A13570 NTR1 agonistML-314 is a brain penetrant nonpeptidic β-arrestin biased ggonist of the neurotensin NTR1 receptor, which exhibits full agonist behavior against NTR1 (EC50 = 2.0 μM) in the primary assay and selectivity against NTR2. Learn More -
JMV 390-1
Catalog No. A16026 JMV 390-1 is a inhibitor of the major neurotensin and neuromedin N degrading enzymes (IC50 values are 31, 40, 52 and 58 nM for endopeptidase 24.15, endopeptidase 24.11, leucine aminopeptidase and endopeptidase 24.16 respectively). Learn More -
SBI-553
Catalog No. A18435 NTR1 allosteric modulatorSBI-553 is a potent and brain penetrant NTR1 allosteric modulator. Learn More