Platelet-Activating Factor (PAF) Receptors

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  1. Aglafoline

    Catalog No. A12257
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    PAF antagonist
    Aglafoline is an effective PAF antagonist not only in vitro, but also in vivo. Learn More
  2. Foropafant

    Catalog No. A13388
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    PAF receptor antagonist
    Foropafant (SR27417) highly potent, competitive, selective and orally active antagonist of platelet-activating factor (PAF) receptor. Learn More
  3. CP-96486

    Catalog No. A12471
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    LTD4/PAF receptor antagonist
    CP-96486 is a potent and orally active leukotriene D4 (LTD4)/platelet activating factor (PAF) receptor antagonist with Kis of 20 and 24 nM, respectively. Learn More
  4. Ginkgolide B

    Catalog No. A10429
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    PAFR antagonist
    Ginkgolide B (BN 52021) is a PAFR antagonist with IC50 of 3.6 μM. Learn More
  5. Ginkgolide A

    Catalog No. A11739
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  6. Rupatadine Fumarate

    Catalog No. A12356
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    PAFR inhibitor/H1 receptor inhibitor
    Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively. Learn More
  7. Rupatadine

    Catalog No. A11222
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    PAFR inhibitor/H1 receptor inhibitor
    Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively. Learn More
  8. Etizolam

    Catalog No. A14257
    PAFR antagonist
    Etizolam is a specific platelet-activating factor (PAF) antagonist with anti-anxiety activity. Learn More
  9. YM-264

    Catalog No. A20139
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    PAF antagonist
    YM-264 is a selective, potent and orally active platelet-activating factor (PAF) antagonist with a pKi value of 8.85 for rabbit platelet membranes. Learn More
  10. 48740 RP

    Catalog No. A12339
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    PAF antagonist
    48740 RP (RP-55778) is a platelet-activating factor (PAF) antagonist. Learn More

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